SCHEMBL7345505

SCHEMBL7345505

COC(=O)C1=C(C)NC(C)=C(C(=O)OCCC2NCc3ccccc32)C1c1cccc(Br)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.55
CACNA1B Q00975 1/20 0.49
ADORA3 P0DMS8 2/20 0.48
CYP1A2 P05177 5/20 0.46
CYP3A4 P08684 5/20 0.46
CYP2C9 P11712 5/20 0.46
CYP2C19 P33261 5/20 0.46
MAPT P10636 5/20 0.46
HIF1A Q16665 4/20 0.46
LMNA P02545 4/20 0.46
CYP2D6 P10635 4/20 0.46
TSHR P16473 4/20 0.46
MEN1 O00255 4/20 0.46
KMT2A Q03164 4/20 0.46
CACNA1C Q13936 3/20 0.46
CACNA1F O60840 2/20 0.46
CACNA1D Q01668 2/20 0.46
CACNA1S Q13698 2/20 0.46
MAPK1 P28482 2/20 0.46
NFKB1 P19838 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7341786 0.90 CACNA1C (0.59) POLBADORA3CYP1A2CYP3A4CYP2C9
SCHEMBL7343716 0.90 CACNA1B (0.49) POLBCACNA1BADORA3CYP1A2CYP3A4
SCHEMBL7349305 0.90 CACNA1B (0.54) POLBCACNA1BADORA3CYP1A2CYP3A4
SCHEMBL7349509 0.87 CACNA1C (0.61) POLBADORA3CYP1A2CYP3A4CYP2C9
SCHEMBL7343611 0.86 CYP1A2 (0.66) POLBADORA3CYP1A2CYP3A4CYP2C9
SCHEMBL7343553 0.86 ADORA3 (0.45) CACNA1BADORA3CYP1A2CYP3A4CYP2C9
SCHEMBL7347767 0.84 CACNA1B (0.49) CACNA1BADORA3CYP1A2CYP3A4CYP2C9
SCHEMBL7344616 0.83 CACNA1B (0.49) POLBCACNA1BADORA3LMNATSHR
SCHEMBL7349531 0.83 ADORA3 (0.55) POLBADORA3CYP1A2CYP3A4CYP2C9
SCHEMBL7348034 0.83 CACNA1C (0.46) CACNA1BADORA3CYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4833150-A HYPOTENSIVES, ANTIARRHYTHMIA AGENTS NELSON RESEARCH & DEVELOPMENT CO. (US) 1989-05-23 US disclosed
US-4652573-A HYPOTENSIVE AGENTS NELSON RESEARCH & DEVELOPMENT CO. (US) 1987-03-24 US disclosed
EP-0194685-A1 1,4-Dihydropyridines Whitby Research Incorporated (US) 1986-09-17 EP disclosed