SCHEMBL7344616

SCHEMBL7344616

COC(=O)C1=C(C)NC(C)=C(C(=O)OCCC2NCc3ccccc32)C1c1ccsc1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 1/20 0.49
ADORA3 P0DMS8 1/20 0.47
KDM4E B2RXH2 6/20 0.46
HSD17B10 Q99714 5/20 0.46
CASP1 P29466 3/20 0.46
HPGD P15428 3/20 0.45
PKM P14618 1/20 0.45
CACNA1F O60840 1/20 0.44
CACNA1D Q01668 1/20 0.44
CACNA1S Q13698 1/20 0.44
CACNA1C Q13936 1/20 0.44
ALDH1A1 P00352 3/20 0.44
CASP7 P55210 2/20 0.44
LMNA P02545 1/20 0.44
ADORA2B P29275 3/20 0.43
TSHR P16473 2/20 0.43
USP2 O75604 1/20 0.43
POLB P06746 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10744175 0.85 ALDH1A1 (0.51) ADORA3KDM4EHSD17B10HPGDPKM
SCHEMBL7349531 0.83 ADORA3 (0.55) ADORA3KDM4EHSD17B10HPGDCACNA1F
SCHEMBL7343553 0.83 ADORA3 (0.45) CACNA1BADORA3KDM4EHSD17B10HPGD
SCHEMBL7348034 0.83 CACNA1C (0.46) CACNA1BADORA3KDM4EHSD17B10HPGD
SCHEMBL7341786 0.83 CACNA1C (0.59) ADORA3CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL7347767 0.83 CACNA1B (0.49) CACNA1BADORA3KDM4EHSD17B10CASP1
SCHEMBL7349305 0.83 CACNA1B (0.54) CACNA1BADORA3KDM4EHSD17B10HPGD
SCHEMBL7343716 0.83 CACNA1B (0.49) CACNA1BADORA3KDM4ECACNA1FCACNA1D
SCHEMBL7345505 0.83 POLB (0.55) CACNA1BADORA3KDM4ECACNA1FCACNA1D
SCHEMBL7342398 0.82 ADORA3 (0.43) CACNA1BADORA3KDM4EHSD17B10HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4833150-A HYPOTENSIVES, ANTIARRHYTHMIA AGENTS NELSON RESEARCH & DEVELOPMENT CO. (US) 1989-05-23 US disclosed
US-4652573-A HYPOTENSIVE AGENTS NELSON RESEARCH & DEVELOPMENT CO. (US) 1987-03-24 US disclosed
EP-0194685-A1 1,4-Dihydropyridines Whitby Research Incorporated (US) 1986-09-17 EP disclosed