SCHEMBL7345522

SCHEMBL7345522

CN1CC2CC(N(C)C(=O)c3nn(C)c4ccccc34)CC(C1)N2C

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.52
CYP3A4 P08684 1/20 0.52
TSHR P16473 1/20 0.52
MAPK1 P28482 1/20 0.52
HSD17B10 Q99714 1/20 0.52
HTR3A P46098 9/20 0.50
HTR3E A5X5Y0 1/20 0.50
SLC22A2 O15244 1/20 0.50
HTR3B O95264 1/20 0.50
CHRNB2 P17787 1/20 0.50
CHRNA3 P32297 1/20 0.50
CHRNA4 P43681 1/20 0.50
KCNH2 Q12809 1/20 0.50
HTR3D Q70Z44 1/20 0.50
HTR3C Q8WXA8 1/20 0.50
SLC47A1 Q96FL8 1/20 0.50
KDM4E B2RXH2 2/20 0.47
RBP4 P02753 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7428799 0.78 ALDH1A1 (0.83) ALDH1A1CYP3A4TSHRMAPK1HSD17B10
SCHEMBL7439648 0.78 ALDH1A1 (0.83) ALDH1A1CYP3A4TSHRMAPK1HSD17B10
SCHEMBL7436275 0.78 HTR3A (0.60) ALDH1A1CYP3A4TSHRMAPK1HSD17B10
SCHEMBL7428794 0.78 ALDH1A1 (0.83) ALDH1A1CYP3A4TSHRMAPK1HSD17B10
SCHEMBL7436272 0.78 HTR3A (0.60) ALDH1A1CYP3A4TSHRMAPK1HSD17B10
SCHEMBL23940247 0.74 KDM4E (0.57) ALDH1A1CYP3A4TSHRMAPK1HSD17B10
SCHEMBL27249478 0.73 ALDH1A1 (0.55) ALDH1A1CYP3A4TSHRMAPK1HSD17B10
SCHEMBL8395556 0.72 HTR3A (0.58) ALDH1A1CYP3A4TSHRMAPK1HSD17B10
Hydrochloric Acid SCHEMBL8400765 0.72 HTR3A (0.57) ALDH1A1CYP3A4TSHRMAPK1HSD17B10
SCHEMBL2087087 0.71 DYRK1A (0.48) ALDH1A1CYP3A4TSHRHSD17B10HTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5344831-A Antiemetics for treatment of nausea from chemotherapy NISSHIN FLOUR MILLING CO., LTD. (JP) 1994-09-06 US disclosed
EP-0558923-A1 Diazabicyclo derivatives as 5-HT3 antagonists NISSHIN FLOUR MILLING CO., LTD. (JP) 1993-09-08 EP disclosed