SCHEMBL7345947

SCHEMBL7345947

CSCC[C@H](NC(=O)N1CCCCCC1)C(=O)N[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)NC(C)(C)C

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 9/20 0.49
YAP1 P46937 3/20 0.49
MME P08473 2/20 0.45
ACE P12821 2/20 0.45
CPA1 P15085 1/20 0.45
ACE2 Q9BYF1 1/20 0.45
MMP9 P14780 1/20 0.44
MMP8 P22894 1/20 0.44
ANPEP P15144 1/20 0.44
DPP7 Q9UHL4 1/20 0.43
CTSL P07711 1/20 0.42
CTSB P07858 1/20 0.42
CTSK P43235 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7340535 0.90 CACNA1B (0.53) CACNA1BYAP1MMEACECPA1
SCHEMBL7347273 0.88 YAP1 (0.53) CACNA1BYAP1MMEACECPA1
SCHEMBL7341833 0.87 CACNA1B (0.62) CACNA1BYAP1MMEACECPA1
SCHEMBL7340850 0.86 TACR2 (0.49) CACNA1BYAP1
SCHEMBL7339047 0.85 YAP1 (0.51) CACNA1BYAP1MMEACECPA1
SCHEMBL7347662 0.83 YAP1 (0.55) CACNA1BYAP1MMEACECPA1
SCHEMBL7344108 0.83 MME (0.51) MMEACECPA1ACE2MMP9
SCHEMBL7339092 0.82 YAP1 (0.60) CACNA1BYAP1MMEACECPA1
SCHEMBL7345875 0.82 YAP1 (0.60) CACNA1BYAP1MMEACECPA1
SCHEMBL7345873 0.82 YAP1 (0.60) CACNA1BYAP1MMEACECPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6423689-B1 Peptidyl calcium channel blockers WARNER-LAMBERT COMPANY 2002-07-23 US disclosed