SCHEMBL7346017

SCHEMBL7346017

CC(C)CC(N)C(=O)NC(Cc1ccc(C#Cc2ccccn2)cc1)C(=O)NC(C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 1/20 0.45
PSMB5 P28074 1/20 0.42
CACNA1B Q00975 2/20 0.41
PTGES O14684 1/20 0.40
AKR1C3 P42330 1/20 0.40
ACACB O00763 7/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7337048 0.89 CACNA1B (0.48) PSMB5CACNA1BACACB
SCHEMBL7338606 0.83 CACNA1B (0.42) CACNA1BACACB
SCHEMBL7346892 0.83 CACNA1B (0.47) PSMB5CACNA1BACACB
SCHEMBL7338188 0.82 KMT2A (0.44) PSMB5CACNA1B
SCHEMBL7346012 0.81 FFAR1 (0.42) FFAR1PTGESAKR1C3ACACB
SCHEMBL7346468 0.79 CACNA1B (0.40) PSMB5CACNA1BACACB
SCHEMBL7343134 0.79 MMP1 (0.52) PSMB5CACNA1B
SCHEMBL7348068 0.79 PSMB5 (0.51) PSMB5CACNA1B
SCHEMBL7338162 0.78 MME (0.56) CACNA1B
SCHEMBL7347212 0.78 FFAR1 (0.45) FFAR1PSMB5CACNA1BACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6423689-B1 Peptidyl calcium channel blockers WARNER-LAMBERT COMPANY 2002-07-23 US claimed
US-6423689-B1 Peptidyl calcium channel blockers WARNER-LAMBERT COMPANY 2002-07-23 US disclosed