SCHEMBL7346806

SCHEMBL7346806

O=C(NCC(NS(=O)(=O)c1ccccc1)C(=O)O)c1cc(OCCCNC2=NCCN2)no1

nearest known ligand 0.61

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 20/20 0.61
ITGAV P06756 17/20 0.61
ITGA2B P08514 17/20 0.52
ITGB5 P18084 1/20 0.46
ITGB6 P18564 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5022907 1.00 ITGB3 (0.61) ITGB3ITGAVITGA2BITGB5ITGB6
SCHEMBL13059981 0.93 ITGB3 (0.54) ITGB3ITGAVITGA2BITGB5ITGB6
SCHEMBL7399998 0.85 ITGB3 (0.51) ITGB3ITGAVITGA2BITGB5ITGB6
SCHEMBL7354623 0.85 ITGB3 (0.58) ITGB3ITGAVITGA2BITGB5
SCHEMBL7347862 0.84 ITGB3 (0.60) ITGB3ITGAVITGA2B
SCHEMBL6111422 0.84 ITGB3 (0.60) ITGB3ITGAVITGA2BITGB5ITGB6
Iodide SCHEMBL7403601 0.84 ITGB3 (0.60) ITGB3ITGAVITGA2BITGB5ITGB6
SCHEMBL5027067 0.84 ITGB3 (0.60) ITGB3ITGAVITGA2BITGB5ITGB6
SCHEMBL7979125 0.83 ITGB3 (0.46) ITGB3ITGAVITGA2B
SCHEMBL7401335 0.81 ITGB3 (0.59) ITGB3ITGAVITGA2BITGB5ITGB6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0828737-A1 ISOXAZOLINE AND ISOXAZOLE DERIVATIVES AS INTEGRIN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-03-18 EP claimed
WO-1996037492-A1 ISOXAZOLINE AND ISOXAZOLE DERIVATIVES AS INTEGRIN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-11-28 WO claimed
US-6214834-B1 ANGIOGENESIS INHIBITORS; ANTIINFLAMMATORY AGENTS; ANTICANCER AGENTS DUPONT PHARMACEUTICALS COMPANY 2001-04-10 US disclosed
WO-1998043962-A1 HETEROCYCLIC INTEGRIN INHIBITOR PRODRUGS DU PONT PHARMACEUTICALS COMPANY (US) 1998-10-08 WO disclosed
EP-0828737-A1 ISOXAZOLINE AND ISOXAZOLE DERIVATIVES AS INTEGRIN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-03-18 EP disclosed
WO-1996037492-A1 ISOXAZOLINE AND ISOXAZOLE DERIVATIVES AS INTEGRIN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-11-28 WO disclosed