SCHEMBL7347323

SCHEMBL7347323

CC(C)(C)N(C[C@@H](O)[C@H](Cc1ccccc1)NC(=O)[C@H](CC(N)=O)NC(=O)c1cc2ccccc2cc1OCc1ccccc1)C(=O)[C@@H]1CCCCN1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.42
ADORA2A P29274 1/20 0.42
ADORA2B P29275 1/20 0.42
ADORA1 P30542 1/20 0.42
CTSD P07339 8/20 0.40
CYP3A4 P08684 3/20 0.40
HTR2B P41595 2/20 0.40
ABCC3 O15438 1/20 0.40
ABCC4 O15439 1/20 0.40
CACNA1F O60840 1/20 0.40
ABCB11 O95342 1/20 0.40
ABCB1 P08183 1/20 0.40
HTR1A P08908 1/20 0.40
DRD2 P14416 1/20 0.40
TACR2 P21452 1/20 0.40
TBXAS1 P24557 1/20 0.40
OPRM1 P35372 1/20 0.40
DRD3 P35462 1/20 0.40
AVPR1A P37288 1/20 0.40
OPRD1 P41143 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9082870 0.89 ADORA3 (0.41) ADORA3ADORA2AADORA2BADORA1CTSD
SCHEMBL7335774 0.85 ADORA3 (0.56) ADORA3ADORA2AADORA2BADORA1CYP3A4
SCHEMBL7267259 0.77 CYP3A4 (0.58) ADORA3ADORA2AADORA2BADORA1CTSD
SCHEMBL9544246 0.76 ADORA3 (0.52) ADORA3ADORA2AADORA2BADORA1CTSD
SCHEMBL9545389 0.75 ADORA3 (0.52) ADORA3ADORA2AADORA2BADORA1REN
SCHEMBL7335261 0.75 CYP3A4 (0.42) ADORA3ADORA2AADORA2BADORA1CTSD
SCHEMBL7268840 0.74 ADORA3 (0.53) ADORA3ADORA2AADORA2BADORA1REN
SCHEMBL9073635 0.73 ADORA3 (0.52) ADORA3ADORA2AADORA2BADORA1CTSD
SCHEMBL7336229 0.72 ADORA3 (0.54) ADORA3ADORA2AADORA2BADORA1CTSD
SCHEMBL9544554 0.72 CYP3A4 (0.52) ADORA3ADORA2AADORA2BADORA1CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0831826-A1 PHARMACEUTICAL COMPOSITION COMPRISING A PROTEINASE INHIBITOR AND A MONOGLYCERIDE F. HOFFMANN-LA ROCHE AG (CH) 1998-04-01 EP disclosed
WO-1996039142-A1 PHARMACEUTICAL COMPOSITION COMPRISING A PROTEINASE INHIBITOR AND A MONOGLYCERIDE F. HOFFMANN-LA ROCHE AG (CH) 1996-12-12 WO disclosed