SCHEMBL9544246

SCHEMBL9544246

CC(C)(C)N(C[C@@H](O)[C@H](Cc1ccccc1)NC(=O)[C@H](CC(N)=O)NC(=O)OCc1ccccc1)C(=O)[C@@H]1C[C@H](Oc2ccccc2)CCN1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.52
ADORA2A P29274 1/20 0.52
ADORA2B P29275 1/20 0.52
ADORA1 P30542 1/20 0.52
PSMB1 P20618 1/20 0.40
CTSL P07711 7/20 0.38
CTSK P43235 5/20 0.38
CTSS P25774 3/20 0.38
PSMB8 P28062 1/20 0.37
PSMB5 P28074 1/20 0.37
BACE1 P56817 3/20 0.37
REN P00797 2/20 0.37
CTSD P07339 1/20 0.37
ITGB3 P05106 2/20 0.37
ITGA2B P08514 2/20 0.37
CAPN1 P07384 1/20 0.36
CTSB P07858 1/20 0.36
ITGAV P06756 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9545389 0.90 ADORA3 (0.52) ADORA3ADORA2AADORA2BADORA1PSMB1
SCHEMBL9073635 0.88 ADORA3 (0.52) ADORA3ADORA2AADORA2BADORA1PSMB1
SCHEMBL7335774 0.88 ADORA3 (0.56) ADORA3ADORA2AADORA2BADORA1PSMB1
SCHEMBL7268840 0.85 ADORA3 (0.53) ADORA3ADORA2AADORA2BADORA1PSMB1
SCHEMBL7336229 0.83 ADORA3 (0.54) ADORA3ADORA2AADORA2BADORA1PSMB1
SCHEMBL9544182 0.81 ADORA3 (0.47) ADORA3ADORA2AADORA2BADORA1BACE1
SCHEMBL9544260 0.80 CTSD (0.42) BACE1CTSD
SCHEMBL9544242 0.80 CYP3A4 (0.42) ADORA3ADORA2AADORA2BADORA1BACE1
SCHEMBL9544557 0.77 CTSD (0.47) CTSD
SCHEMBL7347323 0.76 ADORA3 (0.42) ADORA3ADORA2AADORA2BADORA1PSMB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993018003-A1 SUBSTITUED PIPECOLINIC ACID DERIVATIVES AS HIV PROTEASE INHIBITORS BIO-MEGA/BOEHRINGER INGELHEIM RESEARCH INC. (CA) 1993-09-16 WO claimed