SCHEMBL7347343

SCHEMBL7347343

CN(C)C1CCN(C(=O)c2ccc([N+](=O)[O-])cc2)c2ccccc21

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
OXTR P30559 2/20 0.53
AVPR1A P37288 2/20 0.53
ABCB11 O95342 1/20 0.52
HTR1A P08908 1/20 0.52
CHRM1 P11229 1/20 0.52
AVPR2 P30518 1/20 0.52
SLC6A4 P31645 1/20 0.52
ADRA1A P35348 1/20 0.52
OPRM1 P35372 1/20 0.52
AVPR1B P47901 1/20 0.52
HTT P42858 2/20 0.45
BCHE P06276 1/20 0.44
P2RX4 Q99571 1/20 0.44
KDM4E B2RXH2 1/20 0.44
LMNA P02545 1/20 0.44
MAPT P10636 1/20 0.44
ALDH1A1 P00352 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27314182 1.00 OXTR (0.53) OXTRAVPR1AABCB11HTR1ACHRM1
SCHEMBL4685326 0.93 AVPR1A (0.62) OXTRAVPR1AABCB11HTR1ACHRM1
SCHEMBL7347376 0.89 HTT (0.44) OXTRAVPR1AABCB11HTR1ACHRM1
SCHEMBL7350564 0.85 HTT (0.47) HTTBCHEP2RX4KDM4ELMNA
SCHEMBL7350275 0.84 HTT (0.47) HTTBCHEP2RX4KDM4ELMNA
SCHEMBL7360026 0.83 AVPR1A (0.57) OXTRAVPR1AABCB11HTR1ACHRM1
SCHEMBL27522544 0.83 AVPR1A (0.57) OXTRAVPR1AABCB11HTR1ACHRM1
SCHEMBL7351761 0.81 MAPT (0.46) OXTRAVPR1AABCB11HTR1ACHRM1
SCHEMBL7345512 0.81 KDM4E (0.47) OXTRAVPR1AAVPR2HTTBCHE
SCHEMBL7343913 0.80 AVPR2 (0.56) OXTRAVPR1AABCB11HTR1ACHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1048484-C A process for preparing a composition containing benzoheterocycles OTSUKA PHARMA CO LTD (JP) 2000-01-19 CN disclosed
US-5985869-A USEFUL AS VASODILATORS, HYPOTENSIVE AGENTS, WATER DIURETICS, PLATELET AGGLUTINATION INHIBITORS OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1999-11-16 US disclosed
US-5753677-A Benzoheterocyclic compounds OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed
US-5559230-A VASOPRESSIN ANTAGONISTS, QUINOLINES, BENZAZEPINES, VASODILATION, HYPOTENSIVE AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1996-09-24 US disclosed
EP-0450097-B1 BENZOHETEROCYCLIC COMPOUNDS OTSUKA PHARMA CO LTD (JP) 1996-04-24 EP disclosed
CN-1027505-C Process for preparing benzoheterocyclic compounds OTSUKA PHARMA CO LTD (JP) 1995-01-25 CN disclosed
EP-0450097-A1 BENZOHETEROCYCLIC COMPOUNDS. OTSUKA PHARMA CO LTD (JP) 1991-10-09 EP disclosed
WO-1991005549-A1 BENZOHETEROCYCLIC COMPOUNDS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1991-05-02 WO disclosed