SCHEMBL7360026

SCHEMBL7360026

CN(C)C1CCN(C(=O)c2ccc(N)cc2)c2ccccc21

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 4/20 0.57
OXTR P30559 2/20 0.57
AVPR2 P30518 3/20 0.56
SLC6A4 P31645 3/20 0.56
ABCB11 O95342 1/20 0.56
HTR1A P08908 1/20 0.56
CHRM1 P11229 1/20 0.56
ADRA1A P35348 1/20 0.56
OPRM1 P35372 1/20 0.56
AVPR1B P47901 1/20 0.56
SLC6A2 P23975 2/20 0.44
SLC6A3 Q01959 2/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
KCNH2 Q12809 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27522544 1.00 AVPR1A (0.57) AVPR1AOXTRAVPR2SLC6A4ABCB11
SCHEMBL4681060 0.93 AVPR1A (0.66) AVPR1AOXTRAVPR2SLC6A4ABCB11
SCHEMBL7380286 0.88 AVPR1A (0.49) AVPR1AOXTRAVPR2SLC6A4ABCB11
SCHEMBL7347343 0.83 OXTR (0.53) AVPR1AOXTRAVPR2SLC6A4ABCB11
SCHEMBL27314182 0.83 OXTR (0.53) AVPR1AOXTRAVPR2SLC6A4ABCB11
SCHEMBL7351522 0.83 AVPR1A (0.53) AVPR1AOXTRAVPR2
SCHEMBL7345953 0.82 HSD11B1 (0.51) AVPR1AOXTRAVPR2SLC6A4ABCB11
SCHEMBL7352510 0.82 AVPR1A (0.47) AVPR1AOXTRAVPR2SLC6A4ABCB11
SCHEMBL7345080 0.79 AVPR2 (0.57) AVPR1AOXTRAVPR2SLC6A4ABCB11
SCHEMBL7353739 0.79 AVPR1A (0.57) AVPR1AOXTRAVPR2SLC6A4ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1048484-C A process for preparing a composition containing benzoheterocycles OTSUKA PHARMA CO LTD (JP) 2000-01-19 CN disclosed
US-5985869-A USEFUL AS VASODILATORS, HYPOTENSIVE AGENTS, WATER DIURETICS, PLATELET AGGLUTINATION INHIBITORS OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1999-11-16 US disclosed
US-5753677-A Benzoheterocyclic compounds OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed
US-5559230-A VASOPRESSIN ANTAGONISTS, QUINOLINES, BENZAZEPINES, VASODILATION, HYPOTENSIVE AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1996-09-24 US disclosed
EP-0450097-B1 BENZOHETEROCYCLIC COMPOUNDS OTSUKA PHARMA CO LTD (JP) 1996-04-24 EP disclosed
CN-1027505-C Process for preparing benzoheterocyclic compounds OTSUKA PHARMA CO LTD (JP) 1995-01-25 CN disclosed