SCHEMBL7347666

SCHEMBL7347666

CC(C)CC(N)C(=O)NC(Cc1ccc(CCC(C)(C)C)cc1)C(=O)NC(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 2/20 0.46
PSMB5 P28074 2/20 0.41
PSMB1 P20618 1/20 0.41
PSMB2 P49721 1/20 0.41
MMP1 P03956 4/20 0.40
MMP3 P08254 2/20 0.40
MMP2 P08253 1/20 0.40
NPY4R P50391 6/20 0.39
NPY1R P25929 4/20 0.39
NPY2R P49146 3/20 0.39
NPY5R Q15761 2/20 0.39
MME P08473 1/20 0.39
ACE P12821 1/20 0.39
CPA1 P15085 1/20 0.39
ACE2 Q9BYF1 1/20 0.39
ERAP2 Q6P179 2/20 0.38
ERAP1 Q9NZ08 2/20 0.38
LNPEP Q9UIQ6 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7348068 0.89 PSMB5 (0.51) CACNA1BPSMB5PSMB1PSMB2MMP1
SCHEMBL7337467 0.86 CACNA1B (0.47) CACNA1BPSMB5MMP1MMP3MMP2
SCHEMBL7337635 0.85 CACNA1B (0.41) CACNA1BPSMB5PSMB1PSMB2MMP1
SCHEMBL7343134 0.84 MMP1 (0.52) CACNA1BPSMB5MMP1MMP3MMP2
SCHEMBL7344639 0.84 CACNA1B (0.45) CACNA1BPSMB5PSMB1PSMB2MMP1
SCHEMBL7338188 0.81 KMT2A (0.44) CACNA1BPSMB5PSMB1PSMB2MMP1
SCHEMBL7340728 0.81 CACNA1B (0.48) CACNA1BMMP1MMP3MMP2MME
SCHEMBL7338606 0.81 CACNA1B (0.42) CACNA1BMMP1MMP3MMP2NPY4R
SCHEMBL7337048 0.81 CACNA1B (0.48) CACNA1BPSMB5MMP1MMP3MMP2
SCHEMBL7344645 0.80 MMP1 (0.48) CACNA1BPSMB5MMP1MMP3MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6423689-B1 Peptidyl calcium channel blockers WARNER-LAMBERT COMPANY 2002-07-23 US claimed
US-6423689-B1 Peptidyl calcium channel blockers WARNER-LAMBERT COMPANY 2002-07-23 US disclosed