SCHEMBL7348641

SCHEMBL7348641

C#C[C@H](CC(=O)O)NC(=O)CNC(=O)c1c(F)c(F)cc(NC(=N)N)c1F

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 12/20 0.43
ITGA2B P08514 10/20 0.43
ITGB1 P05556 2/20 0.32
ITGAV P06756 2/20 0.32
ITGA5 P08648 2/20 0.32
MDM4 O15151 1/20 0.32
MDM2 Q00987 1/20 0.32
ITGB5 P18084 1/20 0.31
ITGB6 P18564 1/20 0.31
ITGB8 P26012 1/20 0.31
ITGA8 P53708 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6778246 0.83 FOLH1 (0.32)
SCHEMBL6778874 0.77 ITGB3 (0.51) ITGB3ITGA2BITGB1ITGAVITGA5
SCHEMBL7348656 0.76 CA1 (0.31)
SCHEMBL6773935 0.74 ITGB3 (0.52) ITGB3ITGA2BITGB1ITGAVITGA5
SCHEMBL6777472 0.74 ITGB3 (0.52) ITGB3ITGA2BITGB1ITGAVITGA5
SCHEMBL6773940 0.74 ITGB3 (0.52) ITGB3ITGA2BITGB1ITGAVITGA5
SCHEMBL6783133 0.67 ITGB3 (0.48) ITGB3ITGA2BITGB1ITGAVITGA5
SCHEMBL6783814 0.67 ITGB3 (0.42) ITGB3ITGA2BITGB1ITGAVITGA5
SCHEMBL6776555 0.66 ITGB3 (0.45) ITGB3ITGA2BITGB1ITGAVITGA5
SCHEMBL18553376 0.66 ITGB3 (0.51) ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850221-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1998-07-01 EP claimed
WO-1997008145-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-03-06 WO claimed
EP-0850221-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1998-07-01 EP disclosed
WO-1997008145-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-03-06 WO disclosed