SCHEMBL7348656

SCHEMBL7348656

N=C(N)Nc1cc(F)c(F)c(C(=O)NCC(=O)NC#CCCC(=O)O)c1F

nearest known ligand 0.31

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.31
CA2 P00918 2/20 0.31
CA9 Q16790 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6778880 0.76 CA1 (0.41) CA1CA2
SCHEMBL7348641 0.76 ITGB3 (0.43)
SCHEMBL6778246 0.75 FOLH1 (0.32) CA1CA2CA9
SCHEMBL6773948 0.73 ITGB3 (0.43)
SCHEMBL6783139 0.67 HTT (0.42)
SCHEMBL6776568 0.66 HTT (0.39)
SCHEMBL7340558 0.61 EPHX2 (0.39)
SCHEMBL6783445 0.61 KMT2A (0.40)
SCHEMBL6773426 0.60 MAPK1 (0.45)
SCHEMBL7080325 0.59 ITGB3 (0.64)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850221-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1998-07-01 EP disclosed
WO-1997008145-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-03-06 WO disclosed