SCHEMBL7349059

SCHEMBL7349059

COc1ccc(Cc2cccnc2Cc2ccc(OC)cc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 2/20 0.51
PDE3A Q14432 2/20 0.51
PDE10A Q9Y233 2/20 0.51
LTA4H P09960 1/20 0.50
CYP11B1 P15538 4/20 0.49
CYP11B2 P19099 4/20 0.49
CYP19A1 P11511 1/20 0.49
CYP2C9 P11712 1/20 0.49
RAB9A P51151 3/20 0.48
NPC1 O15118 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.47
LMNA P02545 2/20 0.45
ALDH1A1 P00352 2/20 0.45
CLK4 Q9HAZ1 1/20 0.44
MAPT P10636 1/20 0.43
KDR P35968 2/20 0.43
POLB P06746 1/20 0.42
CYP2D6 P10635 1/20 0.41
ATM Q13315 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ammonia Solution, Strong SCHEMBL15662547 0.98 PDE3B (0.50) PDE3BPDE3APDE10ALTA4HCYP11B1
SCHEMBL28773436 0.91 PDE3B (0.45) PDE3BPDE3APDE10ALTA4HCYP11B1
SCHEMBL10621665 0.90 CYP11B1 (0.50) PDE3BPDE3APDE10ALTA4HCYP11B1
SCHEMBL5382166 0.83 LTA4H (0.55) LTA4HCYP11B1CYP11B2CYP19A1CYP2C9
SCHEMBL23647564 0.82 PDE3B (0.50) PDE3BPDE3APDE10ALTA4HCYP11B1
SCHEMBL4279287 0.82 CYP11B1 (0.50) LTA4HCYP11B1CYP11B2CYP19A1CYP2C9
SCHEMBL9391619 0.82 NPC1 (0.61) LTA4HCYP11B1CYP11B2CYP19A1CYP2C9
SCHEMBL28395651 0.82 RAB9A (0.54) PDE3BPDE3APDE10ALTA4HRAB9A
Ammonia Solution, Strong SCHEMBL29153964 0.80 PDE3B (0.58) PDE3BPDE3APDE10ALTA4HRAB9A
SCHEMBL10625865 0.78 CYP11B1 (0.47) PDE3BPDE3APDE10ALTA4HCYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112292375-B Substituted alkoxypyridinyl indole sulfonamides 优时比制药有限公司 2023-12-05 CN disclosed
CN-110121499-A (aza) indole-, benzothiophene-and benzofuran-3-sulfonamides 优时比制药有限公司 2019-08-13 CN disclosed
CN-109651358-A 4-aminopyridine derivative, its pharmaceutical composition, preparation method and application 上海迪诺医药科技有限公司 2019-04-19 CN disclosed
CN-104755477-B 2-aminopyridine compounds 默克专利股份公司 2017-09-26 CN disclosed
US-4358599-A Synthesis of 4-amino-1,2-hydrocarbyl pyrazolidines via 4-nitro analogs A. H. ROBINS COMPANY, INC. (US) 1982-11-09 US disclosed
US-4309552-A Synthesis of 4-nitro-1,2-hydrocarbyl pyrazolidines and process for preparation thereof A. H. ROBINS COMPANY, INC. (US) 1982-01-05 US disclosed