SCHEMBL7352216

SCHEMBL7352216

C[C@H](COC(=O)c1ccccc1)NC(=O)OC(C)(C)C

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 2/20 0.56
ADRB1 P08588 2/20 0.56
ADRB3 P13945 2/20 0.56
ALDH1A1 P00352 2/20 0.51
PPARA Q07869 4/20 0.50
PPARG P37231 3/20 0.50
SERPINE1 P05121 1/20 0.49
ATM Q13315 1/20 0.49
PPARD Q03181 2/20 0.47
SYK P43405 1/20 0.46
CTSK P43235 3/20 0.46
CTSS P25774 3/20 0.46
MAPK1 P28482 1/20 0.45
HIF1A Q16665 1/20 0.45
TDP1 Q9NUW8 2/20 0.45
HTR1A P08908 1/20 0.45
CYP2D6 P10635 1/20 0.45
SCN1A P35498 1/20 0.45
SLC6A3 Q01959 1/20 0.45
SCN5A Q14524 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7381690 1.00 ADRB2 (0.56) ADRB2ADRB1ADRB3ALDH1A1PPARA
SCHEMBL16648476 1.00 ADRB2 (0.56) ADRB2ADRB1ADRB3ALDH1A1PPARA
SCHEMBL3821539 0.86 PPARA (0.63) ADRB2ADRB1ADRB3ALDH1A1PPARA
SCHEMBL18335299 0.86 PPARA (0.63) ADRB2ADRB1ADRB3ALDH1A1PPARA
SCHEMBL16661377 0.86 ADRB2 (0.53) ADRB2ADRB1ADRB3ALDH1A1PPARA
SCHEMBL4583546 0.83 ATM (0.66) ADRB2ADRB1ADRB3PPARAPPARG
SCHEMBL4583548 0.83 ATM (0.66) ADRB2ADRB1ADRB3PPARAPPARG
SCHEMBL4583537 0.83 ATM (0.66) ADRB2ADRB1ADRB3PPARAPPARG
SCHEMBL10871529 0.82 ATM (0.46) ADRB2ADRB1ADRB3PPARAPPARG
SCHEMBL7485377 0.82 ADRB2 (0.53) ADRB2ADRB1ADRB3ALDH1A1PPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242494-B1 ANGIOGENESIS INHIBITORS, ANTITUMOR AGENTS, DIABETIC RETINOPATHY, AND ANTIINFLAMMATORY AGENTS ABBOTT LABORATORIES 2001-06-05 US disclosed
EP-1073633-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 2001-02-07 EP disclosed
WO-1999057098-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 1999-11-11 WO disclosed