SCHEMBL7352302

SCHEMBL7352302

CC(NC(=O)C(O)[C@H](N)CC1CCCCC1)C(=O)OCc1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 15/20 0.60
METAP1 P53582 7/20 0.60
CTSL P07711 1/20 0.46
CTSB P07858 1/20 0.46
CTSS P25774 1/20 0.46
CTSK P43235 1/20 0.46
REN P00797 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16730492 0.88 METAP2 (0.51) METAP2METAP1
SCHEMBL6476379 0.84 METAP2 (0.64) METAP2METAP1CTSLCTSBCTSS
SCHEMBL6477146 0.83 METAP2 (0.70) METAP2METAP1CTSS
SCHEMBL7353359 0.82 METAP2 (0.78) METAP2METAP1REN
Hydrochloric Acid SCHEMBL7356007 0.81 METAP2 (0.76) METAP2METAP1REN
SCHEMBL7360854 0.81 METAP2 (0.60) METAP2METAP1REN
SCHEMBL1863098 0.80 CTSK (0.57) METAP2METAP1CTSLCTSBCTSS
SCHEMBL8269724 0.80 CTSK (0.57) METAP2METAP1CTSLCTSBCTSS
SCHEMBL1863093 0.80 CTSK (0.57) METAP2METAP1CTSLCTSBCTSS
SCHEMBL1863096 0.80 CTSK (0.57) METAP2METAP1CTSLCTSBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242494-B1 ANGIOGENESIS INHIBITORS, ANTITUMOR AGENTS, DIABETIC RETINOPATHY, AND ANTIINFLAMMATORY AGENTS ABBOTT LABORATORIES 2001-06-05 US claimed
EP-1073633-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 2001-02-07 EP claimed
WO-1999057098-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 1999-11-11 WO claimed
US-6242494-B1 ANGIOGENESIS INHIBITORS, ANTITUMOR AGENTS, DIABETIC RETINOPATHY, AND ANTIINFLAMMATORY AGENTS ABBOTT LABORATORIES 2001-06-05 US disclosed