SCHEMBL7352385

SCHEMBL7352385

O=c1[nH]nc2c(Cl)nc3ccc(Cl)cc3n12

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CUL4A Q13619 1/20 0.48
AHR P35869 1/20 0.45
ADORA1 P30542 2/20 0.40
PDE2A O00408 3/20 0.39
PDE10A Q9Y233 3/20 0.39
PDE3B Q13370 2/20 0.39
PDE3A Q14432 2/20 0.39
PDE5A O76074 1/20 0.39
PDE1A P54750 1/20 0.39
PDE1B Q01064 1/20 0.39
PDE1C Q14123 1/20 0.39
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
GLA P06280 1/20 0.37
POLB P06746 1/20 0.37
GAA P10253 1/20 0.37
HPGD P15428 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5730932 0.79 ADORA1 (0.45) ADORA1
SCHEMBL5429671 0.74 ADORA1 (0.77) ADORA1KDM4EALDH1A1NPSR1
SCHEMBL7418199 0.73 DAO (0.49) ADORA1NPSR1
SCHEMBL5362675 0.73 ADORA3 (0.43) AHRADORA1
SCHEMBL7351886 0.71 PDE5A (0.50) PDE5ANPSR1
SCHEMBL5356006 0.70 ADORA1 (0.52) ADORA1ALDH1A1
SCHEMBL5355187 0.70 ADORA1 (0.52) ADORA1KDM4EALDH1A1GAA
SCHEMBL10846312 0.70 CUL4A (0.54) CUL4APDE2APDE10A
SCHEMBL22432488 0.70 AHR (0.56) AHRKDM4EALDH1A1GAAHSD17B10
SCHEMBL8118931 0.69 CUL4A (0.52) CUL4APDE2APDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0633885-A1 TRIAZOLOQUINOXALIN-1,4-DIONES AND THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1995-01-18 EP disclosed
WO-1993006103-A1 TRIAZOLOQUINOXALIN-1,4-DIONES AND THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1993-04-01 WO disclosed