SCHEMBL5362675

SCHEMBL5362675

O=c1[nH]nc2cnc3ccc(Cl)cc3n12

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.43
ADORA1 P30542 1/20 0.43
CHEK1 O14757 9/20 0.40
NOTUM Q6P988 3/20 0.40
AHR P35869 1/20 0.39
GABRA1 P14867 1/20 0.36
GABRG2 P18507 1/20 0.36
GABRB3 P28472 1/20 0.36
GABRA5 P31644 1/20 0.36
GABRA3 P34903 1/20 0.36
GABRA2 P47869 1/20 0.36
GABRA6 Q16445 1/20 0.36
TLR8 Q9NR97 1/20 0.36
PIK3CB P42338 1/20 0.36
PRKDC P78527 1/20 0.36
ATM Q13315 1/20 0.36
ATR Q13535 1/20 0.36
ATRIP Q8WXE1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5355017 0.82 CHEK1 (0.40) CHEK1NOTUM
SCHEMBL796231 0.82 CHEK1 (0.58) CHEK1GABRA1GABRG2GABRB3GABRA5
SCHEMBL560634 0.78 MAPT (0.54) ADORA3ADORA1CHEK1
SCHEMBL7352385 0.73 CUL4A (0.48) ADORA1AHR
SCHEMBL30978979 0.71 KMO (0.40) NOTUMTLR8
SCHEMBL5350608 0.70 HPGD (0.44) CHEK1
SCHEMBL5468928 0.70 CHEK1 (0.68) CHEK1
SCHEMBL10885012 0.68 PRKDC (0.51) ADORA3ADORA1PIK3CBPRKDCATM
SCHEMBL31612377 0.67 ADORA3 (0.41) ADORA3ADORA1AHRPIK3CBPRKDC
SCHEMBL30231077 0.67 HPGD (0.45) ADORA3ADORA1GABRA1GABRG2GABRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7202245-B2 Substituted 4-amino[1,2,4]triazolo[4,3-a] quinoxalines PFIZER INC. (US) 2007-04-10 US disclosed