SCHEMBL7354464

SCHEMBL7354464

Cc1ccc(NC(=O)C(O)[C@H](N)CC2CCCCC2)cc1

nearest known ligand 0.78

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 18/20 0.78
METAP1 P53582 7/20 0.78
PLAU P00749 1/20 0.51
HPN P05981 1/20 0.51
HTR1E P28566 1/20 0.47
S1PR3 Q99500 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7445063 1.00 METAP2 (0.78) METAP2METAP1PLAUHPNHTR1E
SCHEMBL6484048 0.88 METAP2 (1.00) METAP2METAP1
SCHEMBL7353275 0.87 METAP2 (0.60) METAP2METAP1
SCHEMBL7361364 0.87 METAP2 (0.60) METAP2METAP1
SCHEMBL7362323 0.87 METAP2 (0.60) METAP2METAP1
SCHEMBL7354371 0.87 METAP2 (0.70) METAP2METAP1
SCHEMBL7351136 0.86 METAP2 (0.66) METAP2METAP1
SCHEMBL7357016 0.86 METAP2 (0.60) METAP2METAP1
Hydrochloric Acid SCHEMBL7356659 0.86 METAP2 (0.69) METAP2METAP1
SCHEMBL7358435 0.84 METAP2 (0.57) METAP2METAP1PLAUHPN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242494-B1 ANGIOGENESIS INHIBITORS, ANTITUMOR AGENTS, DIABETIC RETINOPATHY, AND ANTIINFLAMMATORY AGENTS ABBOTT LABORATORIES 2001-06-05 US claimed
EP-1073633-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 2001-02-07 EP claimed
WO-1999057098-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 1999-11-11 WO claimed
US-6242494-B1 ANGIOGENESIS INHIBITORS, ANTITUMOR AGENTS, DIABETIC RETINOPATHY, AND ANTIINFLAMMATORY AGENTS ABBOTT LABORATORIES 2001-06-05 US disclosed
EP-1073633-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 2001-02-07 EP disclosed
WO-1999057098-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 1999-11-11 WO disclosed