SCHEMBL7362323

SCHEMBL7362323

N[C@H](CC1CCCCC1)C(O)C(=O)Nc1ccc(F)cc1

nearest known ligand 0.60

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 15/20 0.60
METAP1 P53582 7/20 0.60
KLK7 P49862 3/20 0.50
USP30 Q70CQ3 1/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6487669 0.88 METAP2 (0.78) METAP2METAP1
SCHEMBL7354464 0.87 METAP2 (0.78) METAP2METAP1
SCHEMBL7353275 0.87 METAP2 (0.60) METAP2METAP1NPC1RAB9A
SCHEMBL7361364 0.87 METAP2 (0.60) METAP2METAP1NPC1RAB9A
SCHEMBL7445063 0.87 METAP2 (0.78) METAP2METAP1
SCHEMBL7354371 0.87 METAP2 (0.70) METAP2METAP1KLK7
SCHEMBL7358435 0.86 METAP2 (0.57) METAP2METAP1
Hydrochloric Acid SCHEMBL7356659 0.86 METAP2 (0.69) METAP2METAP1KLK7
SCHEMBL7351136 0.84 METAP2 (0.66) METAP2METAP1KLK7NPC1RAB9A
SCHEMBL7357016 0.84 METAP2 (0.60) METAP2METAP1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242494-B1 ANGIOGENESIS INHIBITORS, ANTITUMOR AGENTS, DIABETIC RETINOPATHY, AND ANTIINFLAMMATORY AGENTS ABBOTT LABORATORIES 2001-06-05 US claimed
EP-1073633-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 2001-02-07 EP claimed
WO-1999057098-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 1999-11-11 WO claimed
US-6242494-B1 ANGIOGENESIS INHIBITORS, ANTITUMOR AGENTS, DIABETIC RETINOPATHY, AND ANTIINFLAMMATORY AGENTS ABBOTT LABORATORIES 2001-06-05 US disclosed
EP-1073633-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 2001-02-07 EP disclosed
WO-1999057098-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 1999-11-11 WO disclosed