SCHEMBL7354776

SCHEMBL7354776

Cc1nc(CC2CCCCC2)nc(O)c1N

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 2/20 0.46
NOS1 P29475 2/20 0.33
NOS2 P35228 2/20 0.33
CHRM3 P20309 1/20 0.33
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
CHRM4 P08173 1/20 0.32
NOS3 P29474 1/20 0.32
FEN1 P39748 1/20 0.31
TLR7 Q9NYK1 1/20 0.31
NPY5R Q15761 1/20 0.31
RAB9A P51151 2/20 0.31
MEN1 O00255 1/20 0.31
MAPT P10636 1/20 0.31
KMT2A Q03164 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
KDM4E B2RXH2 1/20 0.30
NPC1 O15118 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11348979 0.83 HRH4 (0.44) HRH4NOS1NOS2PDE4APDE4B
SCHEMBL7176775 0.75 HRH4 (0.59) HRH4NOS1NOS2NOS3MEN1
SCHEMBL11348211 0.74 HRH4 (0.35) HRH4
SCHEMBL4419056 0.71 CHRM3 (0.39) HRH4CHRM3PDE4APDE4BPDE4C
SCHEMBL19398339 0.70 MAPT (0.40) MAPT
SCHEMBL18069714 0.68 HRH4 (0.42) HRH4CHRM3PDE4APDE4BPDE4C
SCHEMBL21573227 0.68 HRH4 (0.39) HRH4PDE4APDE4BPDE4CPDE4D
SCHEMBL2118395 0.68 HRH4 (0.39) HRH4PDE4APDE4BPDE4CPDE4D
SCHEMBL15458824 0.67 LMNA (0.39) RAB9AMEN1MAPTKMT2AKDM4E
SCHEMBL15458828 0.67 ASPH (0.38) HRH4PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000027826-A1 NOVEL PYRIMIDINES, THE PRODUCTION THEREOF AND THEIR USE BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-05-18 WO disclosed