SCHEMBL7355569

SCHEMBL7355569

COc1ccccc1C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)OC(C)(C)C)C(C)C

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ELANE P08246 2/20 0.46
CMA1 P23946 11/20 0.45
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
ROCK2 O75116 1/20 0.43
NPC1 O15118 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22209502 0.91 NPC1 (0.46) ELANEMEN1KMT2ANPC1
SCHEMBL18619641 0.91 NPC1 (0.46) ELANEMEN1KMT2ANPC1
SCHEMBL20484718 0.87 MEN1 (0.53) ELANECMA1MEN1KMT2ANPC1
SCHEMBL3177023 0.87 MEN1 (0.53) ELANECMA1MEN1KMT2ANPC1
SCHEMBL8087773 0.83 LMNA (0.50) ELANECMA1MEN1KMT2A
SCHEMBL3470215 0.83 LMNA (0.50) ELANECMA1MEN1KMT2A
SCHEMBL10573052 0.82 ELANE (0.51) ELANECMA1
SCHEMBL714622 0.81 NPC1 (0.46) KMT2ANPC1
SCHEMBL717020 0.81 PREP (0.62)
SCHEMBL717019 0.81 PREP (0.62)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0743953-A1 DIASTEREOMERIC PURE TRIFLUOROMETHYL KETONE PEPTIDE DERIVATIVES AS INHIBITORS OF HUMAN LEUKOCYTE ELASTASE ZENECA LIMITED (GB) 1996-11-27 EP disclosed
WO-1995021855-A1 DIASTEREOMERIC PURE TRIFLUOROMETHYL KETONE PEPTIDE DERIVATIVES AS INHIBITORS OF HUMAN LEUKOCYTE ELASTASE ZENECA LIMITED (GB) 1995-08-17 WO disclosed