SCHEMBL7355802

SCHEMBL7355802

CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C(=O)O)C(C)C

nearest known ligand 0.74

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CTSK P43235 12/20 0.74
CTSB P07858 5/20 0.74
CTSL P07711 6/20 0.67
CTSS P25774 3/20 0.67
CAPN1 P07384 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7355798 1.00 CTSK (0.74) CTSKCTSBCTSLCTSSCAPN1
SCHEMBL29860839 0.92 CTSK (0.70) CTSKCTSBCTSLCTSSCAPN1
SCHEMBL31512934 0.90 CTSK (0.69) CTSKCTSBCTSLCTSSCAPN1
SCHEMBL31512923 0.90 CTSK (0.69) CTSKCTSBCTSLCTSSCAPN1
SCHEMBL6664289 0.90 CTSK (0.67) CTSKCTSBCTSLCTSSCAPN1
SCHEMBL31512942 0.90 CTSK (0.69) CTSKCTSBCTSLCTSSCAPN1
SCHEMBL7275434 0.89 ECE1 (0.65) CTSKCTSBCTSLCTSSCAPN1
SCHEMBL25406813 0.89 CTSK (0.77) CTSKCTSBCTSLCTSSCAPN1
SCHEMBL4872585 0.89 CTSK (0.77) CTSKCTSBCTSLCTSSCAPN1
SCHEMBL20770085 0.89 CTSK (0.77) CTSKCTSBCTSLCTSSCAPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3953463-B1 STABILIZED GLYCOSIDE HYDROLASE VARIANTS NOVOZYMES AS (DK) 2025-08-06 EP disclosed
CN-118530973-A Stabilized cellulase variants 诺维信公司 2024-08-23 CN disclosed
CN-118460512-A Stabilized cellulase variants 诺维信公司 2024-08-09 CN disclosed
CN-112204137-B Stabilized cellulase variants 诺维信公司 2024-05-14 CN disclosed
CN-112272701-B Stabilized cellulase variants 诺维信公司 2024-05-14 CN disclosed
EP-4133066-A1 CARBOHYDRATE BINDING MODULE VARIANTS Novozymes A/S (DK) 2023-02-15 EP disclosed
US-11566239-B2 Stabilized cellulase variants NOVOZYMES A/S (DK) 2023-01-31 US disclosed
CN-115210371-A Carbohydrate binding module variants 诺维信公司 2022-10-18 CN disclosed
US-20220186151-A1 STABILIZED GLYCOSIDE HYDROLASE VARIANTS NOVOZYMES A/S (DK) 2022-06-16 US disclosed
EP-3953463-A1 STABILIZED GLYCOSIDE HYDROLASE VARIANTS Novozymes A/S (DK) 2022-02-16 EP disclosed
WO-1998025949-A1 SUBSTITUTED 5-AMINO-1,3,4-THIADIAZOLE-2-THIONES PROSCRIPT, INC. (US) 1998-06-18 WO disclosed
EP-0845002-A2 AMINO ACID AMIDES OF 5-AMINO-1,3,4-THIADIAZONES AND THEIR USE AS INHIBITORS FOR MATRIX METALLOPROTEINASES PROSCRIPT, INC. (US) 1998-06-03 EP disclosed
US-5677282-A ENZYME INHIBITOR; OSTEOARTHRITIS AND RHEUMATIC DISORDERS PROSCRIPT, INC. (US) 1997-10-14 US disclosed
WO-1996040745-A2 AMINO ACID AMIDES OF 5-AMINO-1,3,4-THIADIAZONES AND THEIR USE AS INHIBITORS FOR MATRIX METALLOPROTEINASES PROSCRIPT, INC. (US) 1996-12-19 WO disclosed