SCHEMBL7356003

SCHEMBL7356003

COC(=O)C(CNC(=O)c1ccc(C(=O)NCCNC(=N)N(C(=O)OC(C)(C)C)C(=O)OC(C)(C)C)s1)Nc1ncccn1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AKT3 Q9Y243 12/20 0.35
ALDH1A1 P00352 1/20 0.31
CYP3A4 P08684 1/20 0.31
MAPT P10636 1/20 0.31
CYP2C9 P11712 1/20 0.31
PKM P14618 1/20 0.31
CYP2C19 P33261 1/20 0.31
SIRT2 Q8IXJ6 1/20 0.31
SIRT1 Q96EB6 1/20 0.31
SIRT3 Q9NTG7 1/20 0.31
ACKR3 P25106 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6502327 0.85 AKT3 (0.35) AKT3
SCHEMBL6502329 0.81 AKT3 (0.35) AKT3SIRT2SIRT1SIRT3
SCHEMBL6502332 0.80 AKT3 (0.33) AKT3MAPTSIRT2SIRT1SIRT3
SCHEMBL7452371 0.76 HPGD (0.52) ALDH1A1MAPTACKR3
SCHEMBL7456483 0.73 ACKR3 (0.43) AKT3ACKR3
SCHEMBL6503512 0.73 SYK (0.41) ALDH1A1
SCHEMBL7453315 0.72 HPGDS (0.37) AKT3ACKR3
SCHEMBL6494160 0.71 GRIN3B (0.41) AKT3
SCHEMBL6494179 0.70 ITGB3 (0.42)
SCHEMBL7456462 0.68 ITGB3 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1091952-A1 THIOPHENE AND FURAN 2,5-DICARBOXAMIDES USEFUL IN THE TREATMENT OF CANCER BIOCHEM PHARMA INC (CA) 2001-04-18 EP disclosed
WO-2000000486-A1 THIOPHENE AND FURAN 2,5-DICARBOXAMIDES USEFUL IN THE TREATMENT OF CANCER BIOCHEM PHARMA INC. (US) 2000-01-06 WO disclosed