SCHEMBL7356284

SCHEMBL7356284

N[C@H](CC1CCCCC1)C(O)C(=O)Nc1cccc(OC(F)(F)F)c1

nearest known ligand 0.61

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 13/20 0.61
METAP1 P53582 6/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7350513 0.99 METAP2 (0.60) METAP2METAP1
SCHEMBL21582918 0.86 METAP2 (0.65) METAP2METAP1
SCHEMBL7355939 0.86 METAP2 (0.65) METAP2METAP1
Hydrochloric Acid SCHEMBL7350300 0.85 METAP2 (0.64) METAP2METAP1
SCHEMBL7358037 0.85 METAP2 (0.70) METAP2METAP1
Hydrochloric Acid SCHEMBL7353872 0.84 METAP2 (0.69) METAP2METAP1
SCHEMBL7362110 0.84 METAP2 (0.65) METAP2METAP1
SCHEMBL7354183 0.84 EPHX2 (0.54) METAP2METAP1
SCHEMBL7360474 0.84 METAP2 (0.66) METAP2METAP1
Hydrochloric Acid SCHEMBL7361219 0.84 METAP2 (0.64) METAP2METAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242494-B1 ANGIOGENESIS INHIBITORS, ANTITUMOR AGENTS, DIABETIC RETINOPATHY, AND ANTIINFLAMMATORY AGENTS ABBOTT LABORATORIES 2001-06-05 US claimed
EP-1073633-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 2001-02-07 EP claimed
WO-1999057098-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 1999-11-11 WO claimed
US-6242494-B1 ANGIOGENESIS INHIBITORS, ANTITUMOR AGENTS, DIABETIC RETINOPATHY, AND ANTIINFLAMMATORY AGENTS ABBOTT LABORATORIES 2001-06-05 US disclosed
EP-1073633-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 2001-02-07 EP disclosed
WO-1999057098-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 1999-11-11 WO disclosed