SCHEMBL7356459

SCHEMBL7356459

Cc1nc2cc(Cl)cc(C(=O)O)c2o1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.42
GPR35 Q9HC97 2/20 0.42
USP2 O75604 1/20 0.42
POLB P06746 1/20 0.42
HPGD P15428 1/20 0.42
ALOX15 P16050 1/20 0.42
ALOX12 P18054 1/20 0.42
CASP1 P29466 1/20 0.42
CASP7 P55210 1/20 0.42
HSD17B10 Q99714 1/20 0.42
KCNH2 Q12809 2/20 0.41
KMT2A Q03164 2/20 0.41
ESR1 P03372 1/20 0.41
MAPT P10636 1/20 0.41
MAPK10 P53779 1/20 0.41
AKR1C4 P17516 1/20 0.40
AKR1C3 P42330 1/20 0.40
AKR1C2 P52895 1/20 0.40
AKR1C1 Q04828 1/20 0.40
NPC1 O15118 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4550751 0.83 ESR2 (0.44) ESR2GPR35KMT2AESR1MAPT
SCHEMBL16047286 0.83 ESR2 (0.47) ESR2USP2POLBHPGDHSD17B10
SCHEMBL2956591 0.77 DHODH (0.61) ESR2POLBESR1MAPTNPC1
SCHEMBL11593571 0.75 KCNA3 (0.37) GPR35USP2POLBHPGDALOX15
SCHEMBL11514237 0.73 GPR35 (0.51) GPR35USP2POLBHPGDALOX15
SCHEMBL1340553 0.73 MAPT (0.63) HPGDHSD17B10KMT2AESR1MAPT
SCHEMBL25083018 0.73 KCNA3 (0.43) ESR2GPR35USP2POLBHSD17B10
SCHEMBL12583782 0.73 KCNH2 (0.55) ESR2POLBKCNH2KMT2AMAPT
SCHEMBL17643040 0.73 MAOB (0.40) ESR2USP2HPGDHSD17B10KMT2A
SCHEMBL11206420 0.70 MAPT (0.44) POLBHPGDALOX15ALOX12HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5726187-A N-alkylpiperidinyl-4-methyl carboxylic esters/amides of condensed ring systems as 5-HT4 receptor antagonists SMITHKLINE BEECHAM PLC (GB) 1998-03-10 US disclosed
EP-0664794-A1 N-ALKYLPIPERIDINYL-4-METHYL CARBOXYLIC ESTERS/AMIDES OF CONDENSED RING SYSTEMS AS 5-HT4 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1995-08-02 EP disclosed
WO-1994008965-A1 N-ALKYLPIPERIDINYL-4-METHYL CARBOXYLIC ESTERS/AMIDES OF CONDENSED RING SYSTEMS AS 5-HT4 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1994-04-28 WO disclosed