SCHEMBL7356591

SCHEMBL7356591

COc1cc(N)c(Cl)cc1C(=O)N(C)OC

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.63
HTR4 Q13639 7/20 0.52
CYP1A2 P05177 2/20 0.52
CYP2D6 P10635 2/20 0.52
HTR3A P46098 2/20 0.52
CYP3A4 P08684 2/20 0.52
CYP2C9 P11712 1/20 0.52
TSHR P16473 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
HTR3E A5X5Y0 1/20 0.51
SLC22A1 O15245 1/20 0.51
HTR3B O95264 1/20 0.51
ALDH1A1 P00352 1/20 0.51
LMNA P02545 1/20 0.51
MPO P05164 1/20 0.51
ADRA2A P08913 1/20 0.51
DRD2 P14416 1/20 0.51
ADRA2C P18825 1/20 0.51
DRD4 P21917 1/20 0.51
HTR2A P28223 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7454538 0.88 GAA (0.67) GAAHTR4CYP1A2CYP2D6HTR3A
SCHEMBL8569184 0.86 GAA (0.44) GAACYP3A4ALDH1A1LMNA
SCHEMBL5925563 0.81 GAA (0.61) GAAHTR4CYP1A2CYP2D6HTR3A
SCHEMBL15651040 0.80 GAA (0.57) GAAHTR4CYP1A2CYP2D6HTR3A
SCHEMBL15651087 0.79 HTR4 (0.56) GAAHTR4CYP1A2CYP2D6HTR3A
SCHEMBL7351910 0.79 GAA (0.73) GAAHTR4CYP1A2CYP2D6HTR3A
SCHEMBL7280230 0.79 GAA (0.73) GAAHTR4CYP1A2CYP2D6HTR3A
SCHEMBL99019 0.79 GAA (0.73) GAAHTR4CYP1A2CYP2D6HTR3A
SCHEMBL725809 0.79 GAA (0.73) GAAHTR4CYP1A2CYP2D6HTR3A
SCHEMBL8572424 0.79 CYP3A4 (0.53) CYP3A4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0700383-B1 NOVEL 1-PHENYLALKANONE 5-HT 4? RECEPTOR LIGANDS SYNTEX INC (US) 1998-09-23 EP disclosed
US-5763458-A NERVOUS SYSTEM DISORDERS, ANXIETY, ANTIDEPRESSANTS AND COGNITION ACTIVATORS SYNTEX (U.S.A.) INC. (US) 1998-06-09 US disclosed
WO-1994027965-A1 NOVEL 1-PHENYLALKANONE 5-HT4 RECEPTOR LIGANDS SYNTEX (U.S.A.) INC. (US) 1994-12-08 WO disclosed