SCHEMBL7357152

SCHEMBL7357152

COc1ccccc1CCNC(=O)C(O)[C@H](N)CC1CCCCC1

nearest known ligand 0.61

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 12/20 0.61
METAP1 P53582 8/20 0.61
HPGD P15428 1/20 0.50
MTNR1A P48039 1/20 0.50
MTNR1B P49286 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7353838 0.99 METAP2 (0.60) METAP2METAP1HPGDMTNR1AMTNR1B
SCHEMBL14984956 0.89 HPGD (0.49) METAP2METAP1HPGDMTNR1AMTNR1B
SCHEMBL12022131 0.86 HPGD (0.47) METAP2METAP1HPGDMTNR1AMTNR1B
SCHEMBL21880703 0.86 HPGD (0.47) METAP2METAP1HPGDMTNR1AMTNR1B
SCHEMBL7350315 0.84 METAP2 (0.77) METAP2METAP1
Hydrochloric Acid SCHEMBL7362199 0.83 METAP2 (0.76) METAP2METAP1
SCHEMBL7353859 0.81 METAP2 (0.65) METAP2METAP1
SCHEMBL7354316 0.81 METAP2 (0.58) METAP2METAP1HPGD
SCHEMBL7361746 0.81 METAP2 (0.64) METAP2METAP1HPGD
Hydrochloric Acid SCHEMBL7361806 0.80 METAP2 (0.63) METAP2METAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242494-B1 ANGIOGENESIS INHIBITORS, ANTITUMOR AGENTS, DIABETIC RETINOPATHY, AND ANTIINFLAMMATORY AGENTS ABBOTT LABORATORIES 2001-06-05 US claimed
EP-1073633-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 2001-02-07 EP claimed
WO-1999057098-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 1999-11-11 WO claimed
US-6242494-B1 ANGIOGENESIS INHIBITORS, ANTITUMOR AGENTS, DIABETIC RETINOPATHY, AND ANTIINFLAMMATORY AGENTS ABBOTT LABORATORIES 2001-06-05 US disclosed
EP-1073633-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 2001-02-07 EP disclosed
WO-1999057098-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 1999-11-11 WO disclosed