SCHEMBL7357763

SCHEMBL7357763

N[C@H](CC1CCCCC1)[C@@H](O)C(=O)NC(CF)C(=O)O

nearest known ligand 0.53

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 12/20 0.53
METAP1 P53582 7/20 0.53
CPB2 Q96IY4 4/20 0.40
MME P08473 1/20 0.40
ACE P12821 1/20 0.40
CPA1 P15085 1/20 0.40
ACE2 Q9BYF1 1/20 0.40
GRN P28799 1/20 0.40
SORT1 Q99523 1/20 0.40
REN P00797 1/20 0.39
LTA4H P09960 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7353581 0.88 METAP2 (0.54) METAP2METAP1CPB2MMEACE
SCHEMBL7357202 0.88 METAP2 (0.54) METAP2METAP1CPB2MMEACE
SCHEMBL7361186 0.84 METAP2 (0.51) METAP2METAP1CPB2REN
SCHEMBL11407267 0.84 METAP2 (0.51) METAP2METAP1CPB2REN
SCHEMBL11407261 0.84 METAP2 (0.51) METAP2METAP1CPB2REN
SCHEMBL7354697 0.84 METAP2 (0.57) METAP2METAP1REN
Hydrochloric Acid SCHEMBL7508388 0.83 METAP2 (0.50) METAP2METAP1CPB2REN
SCHEMBL7361350 0.82 METAP2 (0.61) METAP2METAP1CPB2REN
SCHEMBL7355867 0.82 METAP2 (0.61) METAP2METAP1CPB2REN
Hydrochloric Acid SCHEMBL7358976 0.81 METAP2 (0.60) METAP2METAP1CPB2REN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242494-B1 ANGIOGENESIS INHIBITORS, ANTITUMOR AGENTS, DIABETIC RETINOPATHY, AND ANTIINFLAMMATORY AGENTS ABBOTT LABORATORIES 2001-06-05 US claimed
EP-1073633-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 2001-02-07 EP claimed
WO-1999057098-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 1999-11-11 WO claimed
US-6242494-B1 ANGIOGENESIS INHIBITORS, ANTITUMOR AGENTS, DIABETIC RETINOPATHY, AND ANTIINFLAMMATORY AGENTS ABBOTT LABORATORIES 2001-06-05 US disclosed
EP-1073633-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 2001-02-07 EP disclosed
WO-1999057098-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 1999-11-11 WO disclosed