SCHEMBL7358671

SCHEMBL7358671

COC(=O)CC(NC(=O)CN)c1cccc([N+](=O)[O-])c1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.48
KDM4E B2RXH2 2/20 0.48
LMNA P02545 2/20 0.48
MAPT P10636 2/20 0.48
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
L3MBTL1 Q9Y468 3/20 0.48
HPGD P15428 2/20 0.48
HTT P42858 2/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
CYP26A1 O43174 1/20 0.46
ITGB3 P05106 1/20 0.46
ITGAV P06756 1/20 0.46
ITGA2B P08514 1/20 0.46
ITGB5 P18084 1/20 0.46
ITGB6 P18564 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7168369 0.99 ALDH1A1 (0.48) ALDH1A1KDM4ELMNAMAPTMEN1
SCHEMBL7365092 0.85 ALDH1A1 (0.50) ALDH1A1KDM4ELMNAMAPTMEN1
Hydrochloric Acid SCHEMBL7172679 0.84 ALDH1A1 (0.49) ALDH1A1KDM4ELMNAMAPTMEN1
SCHEMBL10265619 0.84 ALDH1A1 (0.53) ALDH1A1KDM4ELMNAMAPTMEN1
SCHEMBL665809 0.82 CYP26A1 (0.49) ALDH1A1KDM4ELMNAMAPTMEN1
SCHEMBL24036727 0.81 KCNA5 (0.47) ALDH1A1MAPTMEN1KMT2AHTT
SCHEMBL24036731 0.81 WDR5 (0.50) ALDH1A1MEN1KMT2AHPGD
SCHEMBL24036950 0.81 TACR3 (0.39) MAPTMEN1KMT2AL3MBTL1SMN1; SMN2
SCHEMBL665345 0.80 MEN1 (0.51) ALDH1A1LMNAMAPTMEN1KMT2A
SCHEMBL8297473 0.80 MEN1 (0.51) ALDH1A1LMNAMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1153014-A2 BETA-ALANINE DERIVATIVES MERCK PATENT GmbH (DE) 2001-11-14 EP disclosed
WO-2000048996-A2 β-ALANINE DERIVATIVES MERCK PATENT GMBH (DE) 2000-08-24 WO disclosed