SCHEMBL7358955

SCHEMBL7358955

COc1ccc2c(c1)-c1noc(N3CCNCC3)c1CC2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.49
CYP2D6 P10635 2/20 0.49
HTR3E A5X5Y0 2/20 0.43
HTR3B O95264 2/20 0.43
HTR3A P46098 2/20 0.43
HTR3D Q70Z44 2/20 0.43
HTR3C Q8WXA8 2/20 0.43
ADRB1 P08588 3/20 0.42
SIGMAR1 Q99720 3/20 0.42
HTR1A P08908 1/20 0.41
HTR1D P28221 1/20 0.41
HTR1B P28222 1/20 0.41
ALDH1A1 P00352 3/20 0.41
MAPT P10636 2/20 0.41
KDM4E B2RXH2 1/20 0.41
MPI P34949 1/20 0.41
NPY5R Q15761 1/20 0.41
NCF1 P14598 1/20 0.40
NPC1 O15118 2/20 0.39
HPGD P15428 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7355029 0.96 CYP1A2 (0.48) CYP1A2CYP2D6HTR3EHTR3BHTR3A
SCHEMBL7349951 0.79 HRH4 (0.56) HTR1AALDH1A1KDM4ENPC1HPGD
SCHEMBL13202414 0.76 CYP1A2 (0.56) CYP1A2CYP2D6SIGMAR1ALDH1A1MAPT
SCHEMBL7356028 0.75 CYP1A2 (0.55) CYP1A2CYP2D6SIGMAR1ALDH1A1MAPT
SCHEMBL7348643 0.75 CYP1A2 (0.55) CYP1A2CYP2D6SIGMAR1ALDH1A1MAPT
SCHEMBL7350762 0.75 HRH4 (0.52) HTR3AHTR1AALDH1A1KDM4ENCF1
SCHEMBL7350260 0.67 HRH1 (0.55) HTR1AALDH1A1KDM4EHPGDSMN1; SMN2
Hydrochloric Acid SCHEMBL7352883 0.67 CYP1A2 (0.41) CYP1A2CYP2D6HTR3ASIGMAR1ALDH1A1
SCHEMBL13659249 0.66 CYP1A2 (1.00) CYP1A2CYP2D6ALDH1A1MAPTKDM4E
SCHEMBL31649581 0.66 CYP1A2 (0.60) CYP1A2CYP2D6ALDH1A1MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5880121-A SEROTONIN 5HT3 ANTAGONIST, USEFUL FOR TREATING ANXIETY, PHYCHIATRIC DISORDERS, NAUSEA, VOMITING AND DRUG DEPENDENCY HOECHST MARION ROUSSEL INC. (US) 1999-03-09 US disclosed