SCHEMBL7355029

SCHEMBL7355029

COc1ccc2c(c1)-c1noc(N3CCCNCC3)c1CC2

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.48
CYP2D6 P10635 2/20 0.48
CHRNB2 P17787 3/20 0.45
CHRNA4 P43681 3/20 0.45
ALDH1A1 P00352 3/20 0.41
NPC1 O15118 3/20 0.41
RAB9A P51151 3/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
HPGD P15428 2/20 0.41
HTR3A P46098 4/20 0.40
HTR1A P08908 3/20 0.40
HTR2B P41595 3/20 0.40
HTR7 P34969 2/20 0.40
HTR1D P28221 2/20 0.40
MAPT P10636 2/20 0.40
TP53 P04637 2/20 0.40
MAPK1 P28482 2/20 0.40
MEN1 O00255 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7358955 0.96 CYP1A2 (0.49) CYP1A2CYP2D6ALDH1A1NPC1RAB9A
SCHEMBL7350762 0.81 HRH4 (0.52) CHRNB2CHRNA4ALDH1A1SMN1; SMN2HPGD
SCHEMBL7349951 0.75 HRH4 (0.56) ALDH1A1NPC1RAB9ASMN1; SMN2HPGD
SCHEMBL13202414 0.72 CYP1A2 (0.56) CYP1A2CYP2D6ALDH1A1NPC1RAB9A
SCHEMBL7356028 0.71 CYP1A2 (0.55) CYP1A2CYP2D6ALDH1A1NPC1RAB9A
SCHEMBL7348643 0.71 CYP1A2 (0.55) CYP1A2CYP2D6ALDH1A1NPC1RAB9A
SCHEMBL7753896 0.68 CHRNB2 (0.50) CYP1A2CYP2D6CHRNB2CHRNA4HTR3A
SCHEMBL13659249 0.66 CYP1A2 (1.00) CYP1A2CYP2D6ALDH1A1NPC1RAB9A
SCHEMBL12932476 0.65 HTR3A (0.64) CHRNB2CHRNA4HTR3AHTR1AHTR2B
SCHEMBL5237992 0.65 ADRB1 (0.86) CHRNB2CHRNA4HTR3AHTR1AHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5880121-A SEROTONIN 5HT3 ANTAGONIST, USEFUL FOR TREATING ANXIETY, PHYCHIATRIC DISORDERS, NAUSEA, VOMITING AND DRUG DEPENDENCY HOECHST MARION ROUSSEL INC. (US) 1999-03-09 US disclosed