SCHEMBL7359237

SCHEMBL7359237

COc1cccc(COc2cc(N)c(Cl)cc2C(=O)CCC2CCN(CCNS(C)(=O)=O)CC2)c1

nearest known ligand 0.86

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.86
ALDH1A1 P00352 2/20 0.86
CYP3A4 P08684 2/20 0.86
CYP2D6 P10635 2/20 0.86
CYP2C19 P33261 2/20 0.86
KMT2A Q03164 2/20 0.86
TP53 P04637 1/20 0.86
CYP2C9 P11712 1/20 0.75
HTR4 Q13639 1/20 0.75
HTR6 P50406 5/20 0.62
HTR2A P28223 1/20 0.60
HTR2C P28335 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8600555 0.99 MEN1 (0.85) MEN1ALDH1A1CYP3A4CYP2D6CYP2C19
SCHEMBL2946020 0.93 MEN1 (1.00) MEN1ALDH1A1CYP3A4CYP2D6CYP2C19
Hydrochloric Acid SCHEMBL2946335 0.92 MEN1 (0.98) MEN1ALDH1A1CYP3A4CYP2D6CYP2C19
Hydrochloric Acid SCHEMBL8647256 0.90 MEN1 (0.79) MEN1ALDH1A1CYP3A4CYP2D6CYP2C19
SCHEMBL548884 0.86 HTR4 (1.00) MEN1ALDH1A1CYP3A4CYP2D6CYP2C19
Hydrochloric Acid SCHEMBL1078401 0.85 HTR4 (0.98) MEN1ALDH1A1CYP3A4CYP2D6CYP2C19
SCHEMBL7354214 0.85 MEN1 (0.85) MEN1ALDH1A1CYP3A4CYP2D6CYP2C19
Hydrochloric Acid SCHEMBL678966 0.84 HTR4 (0.96) MEN1ALDH1A1CYP3A4CYP2D6CYP2C19
Hydrochloric Acid SCHEMBL7361611 0.84 MEN1 (0.84) MEN1ALDH1A1CYP3A4CYP2D6CYP2C19
Hydrochloric Acid SCHEMBL7354355 0.84 MEN1 (0.84) MEN1ALDH1A1CYP3A4CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1994027965-A1 NOVEL 1-PHENYLALKANONE 5-HT4 RECEPTOR LIGANDS SYNTEX (U.S.A.) INC. (US) 1994-12-08 WO disclosed