SCHEMBL7360425

SCHEMBL7360425

Cc1ccccc1NC(=O)C(O)[C@H](N)CC1CCCCC1

nearest known ligand 0.61

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 15/20 0.61
METAP1 P53582 8/20 0.61
KMT2A Q03164 1/20 0.52
TSHR P16473 1/20 0.50
P2RX7 Q99572 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7361788 0.99 METAP2 (0.60) METAP2METAP1KMT2ATSHRP2RX7
SCHEMBL6477713 0.88 METAP2 (0.72) METAP2METAP1P2RX7
SCHEMBL7351163 0.86 METAP2 (0.59) METAP2METAP1
Hydrochloric Acid SCHEMBL7362241 0.85 METAP2 (0.58) METAP2METAP1
SCHEMBL7359944 0.85 METAP2 (0.61) METAP2METAP1
SCHEMBL14984957 0.85 KMT2A (0.55) METAP2METAP1KMT2ATSHRP2RX7
SCHEMBL7361746 0.85 METAP2 (0.64) METAP2METAP1TSHR
SCHEMBL7351644 0.84 METAP2 (0.54) METAP2METAP1
SCHEMBL19350686 0.83 KMT2A (0.50) METAP2METAP1KMT2ATSHRP2RX7
SCHEMBL12022071 0.83 KMT2A (0.53) METAP2METAP1KMT2ATSHRP2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242494-B1 ANGIOGENESIS INHIBITORS, ANTITUMOR AGENTS, DIABETIC RETINOPATHY, AND ANTIINFLAMMATORY AGENTS ABBOTT LABORATORIES 2001-06-05 US claimed
EP-1073633-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 2001-02-07 EP claimed
WO-1999057098-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 1999-11-11 WO claimed
US-6242494-B1 ANGIOGENESIS INHIBITORS, ANTITUMOR AGENTS, DIABETIC RETINOPATHY, AND ANTIINFLAMMATORY AGENTS ABBOTT LABORATORIES 2001-06-05 US disclosed
EP-1073633-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 2001-02-07 EP disclosed
WO-1999057098-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 1999-11-11 WO disclosed