SCHEMBL7360475

SCHEMBL7360475

COC(=O)c1ccc(OC2CCN(C(=O)OC(C)(C)C)CC2C)cc1OC

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 5/20 0.47
STS P08842 2/20 0.47
ALDH1A1 P00352 1/20 0.46
EPHX2 P34913 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
PDE4A P27815 2/20 0.41
PDE4C Q08493 2/20 0.41
PDE4D Q08499 2/20 0.41
PIK3CD O00329 2/20 0.41
PIK3CA P42336 2/20 0.41
PIK3CB P42338 2/20 0.41
PIK3CG P48736 2/20 0.41
EED O75530 1/20 0.41
RBBP4 Q09028 1/20 0.41
SUZ12 Q15022 1/20 0.41
EZH2 Q15910 1/20 0.41
AEBP2 Q6ZN18 1/20 0.41
GPR119 Q8TDV5 2/20 0.40
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7360121 0.91 PDE4B (0.48) PDE4BSTSALDH1A1EPHX2MEN1
SCHEMBL7477254 0.88 PDE4B (0.51) PDE4BSTSALDH1A1EPHX2MEN1
SCHEMBL30606457 0.85 GPR119 (0.53) PDE4BSTSALDH1A1EPHX2MEN1
SCHEMBL7358039 0.85 GPR119 (0.53) PDE4BSTSALDH1A1EPHX2MEN1
SCHEMBL7475681 0.84 PDE4B (0.52) PDE4BSTSALDH1A1EPHX2PIK3CD
SCHEMBL7403357 0.83 PDE4B (0.47) PDE4BSTSALDH1A1PDE4APDE4C
SCHEMBL3151620 0.79 STS (0.55) PDE4BSTSALDH1A1EPHX2MEN1
SCHEMBL13407853 0.79 GPR119 (0.44) PDE4BSTSALDH1A1GPR119
SCHEMBL7472533 0.79 PARP15 (0.52) STSALDH1A1EPHX2GPR119
SCHEMBL7402370 0.78 PDE4B (0.52) PDE4BSTSALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0805681-A4 TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS MERCK & CO INC (US) 1998-05-06 EP disclosed
EP-0805681-A1 TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 1997-11-12 EP disclosed
WO-1996022775-A1 TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1996-08-01 WO disclosed