SCHEMBL7360957

SCHEMBL7360957

C[C@@H]1CN(C(=O)C(O)[C@H](N)CC2CCCCC2)C[C@H](C)O1

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 11/20 0.44
METAP1 P53582 8/20 0.42
POLB P06746 1/20 0.40
REN P00797 1/20 0.37
CTSS P25774 1/20 0.36
DPP4 P27487 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7357037 1.00 METAP2 (0.44) METAP2METAP1POLBRENCTSS
SCHEMBL7357465 0.80 METAP2 (0.47) METAP2METAP1DPP4
SCHEMBL7352932 0.80 METAP2 (0.47) METAP2METAP1DPP4
SCHEMBL7558136 0.80 METAP2 (0.47) METAP2METAP1DPP4
SCHEMBL10408952 0.73 METAP2 (0.55) METAP2METAP1REN
SCHEMBL8910737 0.71 METAP2 (0.54) METAP2METAP1REN
SCHEMBL5848395 0.71 METAP2 (0.56) METAP2METAP1REN
SCHEMBL5848443 0.71 METAP2 (0.56) METAP2METAP1REN
SCHEMBL7761788 0.71 METAP2 (0.56) METAP2METAP1REN
SCHEMBL10420791 0.71 METAP2 (0.56) METAP2METAP1REN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1073633-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 2001-02-07 EP claimed
WO-1999057098-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 1999-11-11 WO claimed
US-6242494-B1 ANGIOGENESIS INHIBITORS, ANTITUMOR AGENTS, DIABETIC RETINOPATHY, AND ANTIINFLAMMATORY AGENTS ABBOTT LABORATORIES 2001-06-05 US disclosed