SCHEMBL7361018

SCHEMBL7361018

COC(=O)[C@H](Cc1ccc(OCC(=O)OCc2ccccc2)cc1)NC(=O)[C@@H]1CCCN1S(=O)(=O)c1ccc(C)cc1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 3/20 0.55
ITGB1 P05556 4/20 0.51
ITGA5 P08648 2/20 0.51
MMP9 P14780 4/20 0.51
MMP2 P08253 3/20 0.51
FKBP1A P62942 2/20 0.50
ALDH1A1 P00352 1/20 0.48
MMP1 P03956 3/20 0.48
MMP3 P08254 2/20 0.48
MMP7 P09237 2/20 0.48
MMP8 P22894 1/20 0.48
ADAM17 P78536 1/20 0.47
YAP1 P46937 5/20 0.47
RAB9A P51151 1/20 0.47
ITGA2 P17301 1/20 0.46
ITGB7 P26010 1/20 0.46
MMP13 P45452 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7508673 0.98 ITGA4 (0.58) ITGA4ITGB1ITGA5MMP9MMP2
SCHEMBL7353665 0.95 ITGA4 (0.61) ITGA4ITGB1ITGA5MMP9MMP2
SCHEMBL7504392 0.93 ITGA4 (0.59) ITGA4ITGB1ITGA5MMP9MMP2
SCHEMBL7325830 0.90 ITGA4 (0.57) ITGA4ITGB1ITGA5FKBP1AMMP1
SCHEMBL7348048 0.89 ITGB1 (0.53) ITGA4ITGB1ITGA5FKBP1AALDH1A1
SCHEMBL6710599 0.88 ITGA4 (0.54) ITGA4ITGB1ITGA5FKBP1AMMP1
SCHEMBL7446444 0.88 ITGA4 (0.61) ITGA4ITGB1ITGA5FKBP1AALDH1A1
SCHEMBL7070012 0.87 FKBP1A (0.59) ITGA4ITGB1ITGA5MMP9MMP2
SCHEMBL7325073 0.87 ITGA4 (0.56) ITGA4ITGB1ITGA5FKBP1AMMP1
SCHEMBL27668499 0.86 ITGB1 (0.63) ITGA4ITGB1ITGA5MMP9MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001972-A1 SUBSTITUTED PHENYLALANINE TYPE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 Elan Pharmaceuticals, Inc. (US) 2000-05-24 EP claimed
WO-1999006431-A1 SUBSTITUTED PHENYLALANINE TYPE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARMACEUTICALS, INC. (US) 1999-02-11 WO claimed
US-6492421-B1 BINDING VERY LATE ANTIGEN-4; INFLAMMATORY DISEASES SUCH AS ASTHMA, ALZHEIMER'S DISEASE, ATHEROSCLEROSIS, AIDS, DEMENTIA, DIABETES, INFLAMMATORY BOWEL DISEASE, RHEUMATOID ARTHRITIS, TISSUE TRANSPLANTATION, TUMOR METASTASIS, MYOCARDIAL ISCHEMIA ATHENA NEUROSCIENCES, INC. 2002-12-10 US disclosed
EP-1001972-A1 SUBSTITUTED PHENYLALANINE TYPE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 Elan Pharmaceuticals, Inc. (US) 2000-05-24 EP disclosed
WO-1999006431-A1 SUBSTITUTED PHENYLALANINE TYPE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARMACEUTICALS, INC. (US) 1999-02-11 WO disclosed