SCHEMBL7361341

SCHEMBL7361341

Cc1ccc(-c2nc(-c3ccncc3)sc2C(=O)CNC(=O)C(C(N)=O)C2CCCCC2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 11/20 0.42
DBF4 Q9UBU7 11/20 0.42
CCNE1 P24864 2/20 0.41
CDK2 P24941 2/20 0.41
TBK1 Q9UHD2 5/20 0.41
IKBKE Q14164 2/20 0.41
MAPT P10636 2/20 0.36
POLB P06746 1/20 0.36
ALDH1A1 P00352 2/20 0.35
ALOX5 P09917 1/20 0.35
GAA P10253 1/20 0.35
CNR1 P21554 1/20 0.35
MEN1 O00255 1/20 0.35
LMNA P02545 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6807089 0.84 CDC7 (0.42) CDC7DBF4CCNE1CDK2TBK1
SCHEMBL6807084 0.72 CDC7 (0.44) CDC7DBF4CCNE1CDK2TBK1
SCHEMBL6807294 0.61 CDC7 (0.49) CDC7DBF4CCNE1CDK2
SCHEMBL8843252 0.59 EPHX1 (0.53) MAPTALDH1A1
SCHEMBL5271748 0.59 CDC7 (0.69) CDC7DBF4CCNE1CDK2MAPT
SCHEMBL4310703 0.59 MASP2 (0.43)
SCHEMBL14059220 0.59 TBK1 (1.00) TBK1IKBKE
Hydrochloric Acid SCHEMBL8843287 0.58 EPHX1 (0.52) MAPTALDH1A1MEN1KMT2A
SCHEMBL953385 0.58 CDC7 (1.00) CDC7DBF4CCNE1CDK2ALDH1A1
SCHEMBL16113884 0.58 CDC7 (1.00) CDC7DBF4CCNE1CDK2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1159273-A1 COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CATHEPSIN S BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2001-12-05 EP disclosed
WO-2000051998-A1 COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CATHEPSIN S BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2000-09-08 WO disclosed