SCHEMBL7362084

SCHEMBL7362084

N[C@H](CC1CCCCC1)C(O)C(=O)NCc1ccco1

nearest known ligand 0.61

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 10/20 0.61
METAP1 P53582 7/20 0.61
USP2 O75604 1/20 0.46
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
TP53 P04637 1/20 0.44
POLB P06746 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7361849 0.99 METAP2 (0.60) METAP2METAP1USP2CYP1A2CYP2C9
SCHEMBL7355924 0.80 METAP2 (0.60) METAP2METAP1USP2POLBKMT2A
Hydrochloric Acid SCHEMBL7355919 0.79 METAP2 (0.59) METAP2METAP1POLBKMT2A
SCHEMBL7354275 0.78 METAP2 (0.63) METAP2METAP1
SCHEMBL7362423 0.78 METAP2 (0.63) METAP2METAP1KMT2A
SCHEMBL7356888 0.77 METAP2 (0.69) METAP2METAP1KMT2A
SCHEMBL7351848 0.77 METAP2 (0.69) METAP2METAP1POLB
SCHEMBL7351333 0.77 METAP2 (0.69) METAP2METAP1POLB
Hydrochloric Acid SCHEMBL7352923 0.77 METAP2 (0.62) METAP2METAP1KMT2A
Hydrochloric Acid SCHEMBL7359791 0.76 METAP2 (0.67) METAP2METAP1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1073633-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 2001-02-07 EP claimed
WO-1999057098-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 1999-11-11 WO claimed
US-6242494-B1 ANGIOGENESIS INHIBITORS, ANTITUMOR AGENTS, DIABETIC RETINOPATHY, AND ANTIINFLAMMATORY AGENTS ABBOTT LABORATORIES 2001-06-05 US disclosed
EP-1073633-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 2001-02-07 EP disclosed
WO-1999057098-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 1999-11-11 WO disclosed