SCHEMBL7362202

SCHEMBL7362202

NC(=O)c1ccc(-c2nn(Cc3ccccc3)c(=O)c3ncccc23)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.54
NPSR1 Q6W5P4 3/20 0.52
CYP1A2 P05177 2/20 0.52
CYP3A4 P08684 2/20 0.52
CYP2C9 P11712 2/20 0.52
CYP2C19 P33261 2/20 0.52
ENPP1 P22413 1/20 0.47
F2RL3 Q96RI0 1/20 0.47
LMNA P02545 2/20 0.47
CYP2D6 P10635 2/20 0.47
HTT P42858 1/20 0.47
PDE4A P27815 3/20 0.47
PDE4B Q07343 3/20 0.47
PDE4C Q08493 3/20 0.47
PDE4D Q08499 3/20 0.47
PDE3B Q13370 1/20 0.44
PDE3A Q14432 1/20 0.44
RORC P51449 1/20 0.44
PSMB1 P20618 1/20 0.44
PSMB5 P28074 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7367921 0.93 PDE4A (0.53) ALDH1A1NPSR1CYP1A2CYP3A4CYP2C9
SCHEMBL7365377 0.91 PDE4A (0.54) ALDH1A1NPSR1CYP1A2CYP3A4CYP2C9
SCHEMBL7365466 0.91 ALDH1A1 (0.56) ALDH1A1NPSR1CYP1A2CYP3A4CYP2C9
SCHEMBL7369761 0.87 ALDH1A1 (0.70) ALDH1A1NPSR1CYP1A2CYP3A4CYP2C9
SCHEMBL7363597 0.86 ALDH1A1 (0.51) ALDH1A1NPSR1CYP1A2CYP3A4CYP2C9
SCHEMBL7367645 0.86 F2RL3 (0.55) ALDH1A1NPSR1CYP1A2CYP3A4CYP2C9
SCHEMBL7361314 0.85 TBXAS1 (0.46) PDE4APDE4BPDE4CPDE4DALOX15
SCHEMBL7368362 0.85 PDE4A (0.54) ALDH1A1NPSR1CYP1A2CYP3A4CYP2C9
SCHEMBL7366591 0.84 ALDH1A1 (0.59) ALDH1A1NPSR1CYP1A2CYP3A4CYP2C9
SCHEMBL7366350 0.84 PDE4A (0.64) ALDH1A1NPSR1CYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5716954-A ANTIINFLAMMATORY AGENT, ANTIHISTAMINES, IMMUNOSUPPRESSION,AUTOIMMUNE DISEASES SYNTEX U.S.A. INC. (US) 1998-02-10 US disclosed
EP-0612321-A1 PYRIDO PYRIDAZINONE AND PYRIDAZINTHIONE COMPOUNDS WITH PDE IV INHIBITING ACTIVITY SYNTEX (U.S.A.) INC. (US) 1994-08-31 EP disclosed
WO-1993007146-A1 BENZO AND PYRIDO PYRIDAZINONE AND PYRIDAZINTHIONE COMPOUNDS WITH PDE IV INHIBITING ACTIVITY SYNTEX (U.S.A.) INC. (US) 1993-04-15 WO disclosed