SCHEMBL7362212

SCHEMBL7362212

O=c1c2ccccc2c(-c2cccc([N+](=O)[O-])c2)nn1Cc1ccccc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.68
PDE4A P27815 3/20 0.66
PDE4B Q07343 2/20 0.66
PDE4C Q08493 2/20 0.66
PDE4D Q08499 2/20 0.66
NPSR1 Q6W5P4 3/20 0.59
CYP1A2 P05177 2/20 0.59
CYP3A4 P08684 2/20 0.59
CYP2C9 P11712 2/20 0.59
CYP2C19 P33261 2/20 0.59
LMNA P02545 2/20 0.59
CYP2D6 P10635 1/20 0.59
HTT P42858 1/20 0.59
CFTR P13569 6/20 0.57
L3MBTL1 Q9Y468 1/20 0.55
RXFP1 Q9HBX9 1/20 0.53
ENPP1 P22413 1/20 0.50
KMT2A Q03164 3/20 0.49
MEN1 O00255 2/20 0.49
POLB P06746 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7369620 0.90 PDE4A (0.61) ALDH1A1PDE4APDE4BPDE4CPDE4D
SCHEMBL7361489 0.87 PDE4D (0.74) ALDH1A1PDE4APDE4BPDE4CPDE4D
SCHEMBL7363642 0.87 PDE4A (0.87) ALDH1A1PDE4APDE4BPDE4CPDE4D
SCHEMBL7368621 0.82 ALDH1A1 (1.00) ALDH1A1PDE4APDE4BPDE4CPDE4D
SCHEMBL7363261 0.82 ALDH1A1 (0.77) ALDH1A1PDE4APDE4BPDE4CPDE4D
SCHEMBL24000529 0.81 ALDH1A1 (0.75) ALDH1A1PDE4APDE4BPDE4CPDE4D
SCHEMBL22721890 0.81 ALDH1A1 (0.75) ALDH1A1PDE4APDE4BPDE4CPDE4D
SCHEMBL29539593 0.81 ALDH1A1 (0.75) ALDH1A1PDE4APDE4BPDE4CPDE4D
SCHEMBL7364068 0.80 PDE4A (0.85) ALDH1A1PDE4APDE4BPDE4CPDE4D
Pyridopyridazinone SCHEMBL6637552 0.80 PDE4A (1.00) ALDH1A1PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5716954-A ANTIINFLAMMATORY AGENT, ANTIHISTAMINES, IMMUNOSUPPRESSION,AUTOIMMUNE DISEASES SYNTEX U.S.A. INC. (US) 1998-02-10 US disclosed
EP-0612321-A1 PYRIDO PYRIDAZINONE AND PYRIDAZINTHIONE COMPOUNDS WITH PDE IV INHIBITING ACTIVITY SYNTEX (U.S.A.) INC. (US) 1994-08-31 EP disclosed
WO-1993007146-A1 BENZO AND PYRIDO PYRIDAZINONE AND PYRIDAZINTHIONE COMPOUNDS WITH PDE IV INHIBITING ACTIVITY SYNTEX (U.S.A.) INC. (US) 1993-04-15 WO disclosed