SCHEMBL7362624

SCHEMBL7362624

CCOC(COc1ccc(CBr)cc1)OCC

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NQO1 P15559 1/20 0.40
PPARA Q07869 6/20 0.39
TDP1 Q9NUW8 2/20 0.35
KDM4E B2RXH2 1/20 0.35
MAPK1 P28482 1/20 0.35
TSHR P16473 1/20 0.34
PPARG P37231 4/20 0.34
PPARD Q03181 3/20 0.34
FFAR1 O14842 2/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28135784 0.86 NQO1 (0.38) NQO1PPARATDP1PPARGKMT2A
SCHEMBL17400983 0.85 NQO1 (0.43) NQO1PPARATDP1MEN1KMT2A
SCHEMBL9828840 0.84 NQO1 (0.39) NQO1PPARATDP1KDM4EMAPK1
SCHEMBL17400969 0.83 NQO1 (0.61) NQO1TDP1KDM4ETSHR
SCHEMBL2140259 0.82 PPARA (0.42) NQO1PPARATSHRPPARGPPARD
SCHEMBL2329778 0.81 KDM4E (0.46) NQO1PPARATDP1KDM4EMAPK1
SCHEMBL16519363 0.81 NQO1 (0.46) NQO1TDP1KDM4ETSHR
SCHEMBL5779539 0.79 USP2 (0.45) NQO1PPARAKDM4ETSHRPPARG
SCHEMBL1951190 0.79 CYP2C9 (0.50) NQO1KDM4EMAPK1TSHRMEN1
SCHEMBL1244852 0.79 CYP4F2 (0.42) PPARAMAPK1PPARGMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0236307-B1 ANTIHYPERTENSIVE AGENTS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THE PREPARATION OF THE AGENTS AND COMPOSITIONS SCHERING CORPORATION (US) 1991-04-17 EP disclosed
US-4840772-A KIT WITH CONTAINERS OF AGENT TO REDUCE INTRAOCULAR PRESSURE AND ANTIINFLAMMATORY STEROID OR BETA-BLOCKER SCHERING CORPORATION (US) 1989-06-20 US disclosed
US-4783444-A SUBSTITUTED DIPEPTIDES SCHERING CORPORATION (US) 1988-11-08 US disclosed
EP-0236307-A1 ANTIHYPERTENSIVE AGENTS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THE PREPARATION OF THE AGENTS AND COMPOSITIONS. SCHERING CORP (US) 1987-09-16 EP disclosed
US-4691049-A Process for preparing a specific diastereomer of a monoamino dicarboxylic acid ester SCHERING CORPORATION (US) 1987-09-01 US disclosed
WO-1987001707-A1 ANTIHYPERTENSIVE AGENTS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THE PREPARATION OF THE AGENTS AND COMPOSITIONS SCHERING CORPORATION (US) 1987-03-26 WO disclosed
US-4584285-A Antihypertensive agents SCHERING CORPORATION (US) 1986-04-22 US disclosed