SCHEMBL736278

SCHEMBL736278

CC(N)c1ccccc1.C[C@@H](Nc1ccc(C(F)(F)F)c(Cl)c1)C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CASR P41180 1/20 0.42
MAPT P10636 2/20 0.40
KDM4E B2RXH2 2/20 0.40
PDE2A O00408 1/20 0.40
GAA P10253 1/20 0.40
MAPK1 P28482 1/20 0.40
RAB9A P51151 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
RAPGEF3 O95398 3/20 0.39
AKR1C3 P42330 1/20 0.38
AKR1C2 P52895 1/20 0.38
SLC1A3 P43003 1/20 0.38
SLC1A2 P43004 1/20 0.38
SLC1A1 P43005 1/20 0.38
CXCR2 P25025 1/20 0.38
KDR P35968 1/20 0.37
RAPGEF4 Q8WZA2 1/20 0.37
PDK1 Q15118 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL733551 0.90 KDR (0.44) CASRMAPTKDM4EPDE2AGAA
SCHEMBL733552 0.90 KDR (0.44) CASRMAPTKDM4EPDE2AGAA
SCHEMBL1555740 0.90 KDR (0.44) CASRMAPTKDM4EPDE2AGAA
Phenethylamine SCHEMBL1846723 0.84 MMP7 (0.41) CASRMAPTKDM4EGAAMAPK1
SCHEMBL1555612 0.79 KDR (0.59) CASRMAPTGAARAB9ANPSR1
SCHEMBL734816 0.79 KDR (0.59) CASRMAPTGAARAB9ANPSR1
SCHEMBL1555605 0.78 SMN1; SMN2 (0.43) MAPTKDM4EMAPK1RAB9ANPSR1
SCHEMBL19951698 0.78 SMN1; SMN2 (0.43) MAPTKDM4EMAPK1RAB9ANPSR1
SCHEMBL735574 0.75 EPHX2 (0.46) KDM4EMAPK1AKR1C3AKR1C2SMN1; SMN2
SCHEMBL11329660 0.74 RAPGEF3 (0.45) CASRMAPTGAANPSR1RAPGEF3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138175-B2 Heterocyclyl compounds HOFFMANN-LA ROCHE INC. (US) 2012-03-20 US disclosed