SCHEMBL7362783

SCHEMBL7362783

COC(=O)/C=C(/C=C/c1ccc(C#N)cc1)c1cccc(C#N)c1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
P4HB P07237 9/20 0.50
MAPT P10636 3/20 0.50
ALDH1A1 P00352 2/20 0.50
LMNA P02545 2/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
MAOB P27338 2/20 0.45
MAOA P21397 1/20 0.45
HDAC2 Q92769 1/20 0.44
ABCG2 Q9UNQ0 1/20 0.43
ESR1 P03372 1/20 0.42
ACHE P22303 1/20 0.42
NPC1 O15118 1/20 0.41
HTT P42858 1/20 0.41
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7362784 1.00 P4HB (0.50) P4HBMAPTALDH1A1LMNAL3MBTL1
SCHEMBL7363691 0.92 P4HB (0.60) P4HBMAOBMAOA
SCHEMBL7363693 0.92 P4HB (0.60) P4HBMAOBMAOA
SCHEMBL7358440 0.88 MAPT (0.50) P4HBMAPTALDH1A1LMNAMAOB
SCHEMBL7358436 0.88 MAPT (0.50) P4HBMAPTALDH1A1LMNAMAOB
SCHEMBL7365006 0.88 P4HB (0.56) P4HBMAOBMAOA
SCHEMBL7365009 0.88 P4HB (0.56) P4HBMAOBMAOA
SCHEMBL7368327 0.87 P4HB (0.52) P4HBMAPTALDH1A1LMNAL3MBTL1
SCHEMBL7368330 0.87 P4HB (0.52) P4HBMAPTALDH1A1LMNAL3MBTL1
SCHEMBL7360197 0.86 MAPT (0.49) MAPTALDH1A1LMNAL3MBTL1MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0892780-B1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS BRISTOL MYERS SQUIBB PHARMA CO (US) 2002-11-20 EP disclosed
US-5942544-A α-branched anilines, toluenes, and analogs thereof as factor Xa inhibitors DUPONT PHARMACEUTICALS COMPANY (US) 1999-08-24 US disclosed
EP-0892780-A1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1999-01-27 EP disclosed
WO-1997030971-A1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-08-28 WO disclosed