SCHEMBL7368330

SCHEMBL7368330

COC(=O)C=C(C=Cc1ccc(C#N)cc1)c1ccc(C#N)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P4HB P07237 4/20 0.52
MAPT P10636 3/20 0.50
ALDH1A1 P00352 2/20 0.50
HDAC2 Q92769 2/20 0.50
LMNA P02545 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
CA12 O43570 2/20 0.45
CA1 P00915 2/20 0.45
CA2 P00918 2/20 0.45
CA9 Q16790 2/20 0.45
TYR P14679 1/20 0.45
CA7 P43166 1/20 0.45
CA14 Q9ULX7 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.44
SNCA P37840 2/20 0.43
HTT P42858 1/20 0.43
GPR183 P32249 1/20 0.43
MAOB P27338 2/20 0.41
MAOA P21397 1/20 0.41
PTPN1 P18031 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7368327 1.00 P4HB (0.52) P4HBMAPTALDH1A1HDAC2LMNA
SCHEMBL7362783 0.87 P4HB (0.50) P4HBMAPTALDH1A1HDAC2LMNA
SCHEMBL7362784 0.87 P4HB (0.50) P4HBMAPTALDH1A1HDAC2LMNA
SCHEMBL7365006 0.87 P4HB (0.56) P4HBMAOBMAOA
SCHEMBL7365009 0.87 P4HB (0.56) P4HBMAOBMAOA
SCHEMBL7102972 0.84 CA12 (0.64) P4HBMAPTALDH1A1HDAC2LMNA
SCHEMBL7102981 0.84 CA12 (0.64) P4HBMAPTALDH1A1HDAC2LMNA
SCHEMBL7360203 0.81 MAPT (0.49) MAPTALDH1A1LMNAL3MBTL1HTT
SCHEMBL7360197 0.81 MAPT (0.49) MAPTALDH1A1LMNAL3MBTL1HTT
SCHEMBL13114501 0.80 HDAC2 (0.68) P4HBMAPTALDH1A1HDAC2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5942544-A α-branched anilines, toluenes, and analogs thereof as factor Xa inhibitors DUPONT PHARMACEUTICALS COMPANY (US) 1999-08-24 US disclosed
EP-0892780-A1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1999-01-27 EP disclosed
WO-1997030971-A1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-08-28 WO disclosed