SCHEMBL7362786

SCHEMBL7362786

CCOC(=O)CCN1CC(=O)N(C2CCCCC2)c2ccc([N+](=O)[O-])cc2C1=O

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.41
MAPK1 P28482 1/20 0.41
CASP3 P42574 2/20 0.40
MAPT P10636 3/20 0.39
TDP1 Q9NUW8 1/20 0.38
LMNA P02545 1/20 0.38
POLB P06746 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
FKBP1A P62942 1/20 0.38
AR P10275 1/20 0.38
KDM4E B2RXH2 1/20 0.38
TSHR P16473 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C19 P33261 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7332949 0.86 ALDH1A1 (0.44) ALDH1A1MAPK1MAPTLMNASMN1; SMN2
SCHEMBL7324337 0.85 CASP1 (0.46) ALDH1A1MAPK1CASP3MAPTTDP1
SCHEMBL7393832 0.83 ALDH1A1 (0.43) ALDH1A1MAPK1CASP3MAPTTDP1
SCHEMBL7539270 0.82 MAPT (0.41) ALDH1A1MAPK1CASP3MAPTLMNA
SCHEMBL7335912 0.82 MAPT (0.41) ALDH1A1MAPK1CASP3MAPTTDP1
SCHEMBL7353647 0.81 MAPT (0.39) ALDH1A1MAPK1CASP3MAPTTDP1
SCHEMBL7327319 0.78 BRD4 (0.41) ALDH1A1MAPK1MAPTTSHR
SCHEMBL7321430 0.78 BRD4 (0.41) ALDH1A1MAPK1TSHR
SCHEMBL3797765 0.77 MAPT (0.47) ALDH1A1MAPK1MAPTTDP1LMNA
SCHEMBL7324527 0.77 MAOB (0.41) ALDH1A1MAPK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5674863-A BENZODIAZEPINEDIONE DERIVATIVE; FIBRINOGIN BINDING INHIBITOR GENENTECH, INC. (US) 1997-10-07 US disclosed
US-5674865-A BENZODIAZEPINEDIONE DERIVATIVE; FIBRINOGIN BINDING INHIBITOR GENENTECH, INC. (US) 1997-10-07 US disclosed
US-5565449-A PLATELET AGGREGATION INHIBITORS GENENTECH, INC. (US) 1996-10-15 US disclosed
EP-0610334-B1 NONPEPTIDYL INTEGRIN INHIBITORS HAVING SPECIFICITY FOR THE GPII B III A RECEPTOR GENENTECH INC (US) 1996-01-24 EP disclosed
WO-1993008174-A1 NONPEPTIDYL INTEGRIN INHIBITORS HAVING SPECIFICITY FOR THE GPIIbIIIa RECEPTOR GENENTECH, INC. (US) 1993-04-29 WO disclosed