SCHEMBL7362989

SCHEMBL7362989

CN[C@@H](COCc1ccccc1)C(=O)OC(C)(C)C

nearest known ligand 0.65

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 2/20 0.65
CTSS P25774 1/20 0.58
PPARG P37231 1/20 0.56
KLK7 P49862 2/20 0.51
KLK5 Q9Y337 2/20 0.51
ITGA4 P13612 1/20 0.48
ITGB7 P26010 1/20 0.48
FOLH1 Q04609 1/20 0.47
SYK P43405 1/20 0.46
MMP9 P14780 1/20 0.45
MMP14 P50281 1/20 0.45
POLB P06746 1/20 0.45
MAPT P10636 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
RAB9A P51151 1/20 0.45
MME P08473 1/20 0.44
CA1 P00915 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9470479 0.87 PPARA (0.67) PPARACTSSPPARGKLK7KLK5
SCHEMBL8070441 0.85 PPARA (0.56) PPARACTSSPPARGKLK7KLK5
SCHEMBL13844843 0.85 PPARA (0.53) PPARACTSSPPARGFOLH1MMP9
SCHEMBL20804457 0.85 PPARA (0.53) PPARACTSSPPARGFOLH1MMP9
SCHEMBL1414148 0.85 PPARA (0.53) PPARACTSSPPARGFOLH1MMP9
Hydrochloric Acid SCHEMBL31612159 0.84 PPARA (0.52) PPARACTSSPPARGFOLH1MMP9
Hydrochloric Acid SCHEMBL1414145 0.84 PPARA (0.52) PPARACTSSPPARGFOLH1MMP9
SCHEMBL19945248 0.84 ITGA4 (0.61) CTSSKLK5ITGA4ITGB7MMP9
SCHEMBL19945249 0.84 ITGA4 (0.61) CTSSKLK5ITGA4ITGB7MMP9
SCHEMBL17817736 0.83 PPARA (0.61) PPARACTSSPPARGFOLH1MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1171116-A N-substituted glycine derivatives as factor Xa inhibitors CORVAS INT INC (US) 1998-01-21 CN disclosed
EP-0801654-A1 N-SUBSTITUTED GLYCINE DERIVATIVES AS INHIBITORS OF FACTOR Xa CORVAS INTERNATIONAL, INC. (US) 1997-10-22 EP disclosed
WO-1996019493-A1 N-SUBSTITUTED GLYCINE DERIVATIVES AS INHIBITORS OF FACTOR Xa CORVAS INTERNATIONAL, INC. (US) 1996-06-27 WO disclosed