SCHEMBL7363588

SCHEMBL7363588

CC(C)Cc1nc(-c2cccnc2)oc1C(=O)C(CCNC(=O)CC(C)(C)CC(N)=O)c1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.37
KDM4E B2RXH2 8/20 0.37
HPGD P15428 5/20 0.37
HSD17B10 Q99714 5/20 0.37
RAB9A P51151 3/20 0.37
NPC1 O15118 3/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
TP53 P04637 1/20 0.37
TSHR P16473 1/20 0.37
PPARG P37231 3/20 0.37
PPARA Q07869 3/20 0.37
EPHX2 P34913 2/20 0.35
POLB P06746 3/20 0.34
USP2 O75604 1/20 0.34
ESR1 P03372 1/20 0.34
IKBKB O14920 1/20 0.33
CTSL P07711 1/20 0.33
CTSS P25774 1/20 0.33
CTSK P43235 1/20 0.33
PDE10A Q9Y233 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6801355 0.71 CTSL (0.38) ALDH1A1KDM4EHPGDHSD17B10RAB9A
SCHEMBL6801357 0.69 CTSL (0.42) ALDH1A1KDM4EHPGDHSD17B10RAB9A
SCHEMBL6807134 0.68 CTSL (0.44) PPARGPPARAPOLBCTSL
SCHEMBL6807131 0.67 PPARG (0.38) ALDH1A1KDM4EHPGDHSD17B10RAB9A
SCHEMBL6800330 0.66 AAK1 (0.45) ALDH1A1KDM4EHPGDHSD17B10RAB9A
SCHEMBL6800322 0.65 KDM4E (0.38) ALDH1A1KDM4EHPGDHSD17B10RAB9A
SCHEMBL7365739 0.64 ERCC1 (0.36) ALDH1A1HPGDSMN1; SMN2EPHX2MAPK1
SCHEMBL6797431 0.63 TP53 (0.35) TP53PPARGPPARACTSL
SCHEMBL7366743 0.61 LMNA (0.41) ALDH1A1KDM4ERAB9ANPC1SMN1; SMN2
SCHEMBL6797434 0.61 CTSL (0.37) TP53PPARGPPARACTSLCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1159273-A1 COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CATHEPSIN S BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2001-12-05 EP disclosed
WO-2000051998-A1 COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CATHEPSIN S BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2000-09-08 WO disclosed