SCHEMBL7363752

SCHEMBL7363752

COC(=O)CC(CN)c1ccc(OC)c(OC)c1

nearest known ligand 0.59

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.59
TNF P01375 10/20 0.53
PDE4A P27815 5/20 0.53
PDE4B Q07343 5/20 0.53
PDE4C Q08493 5/20 0.53
PDE4D Q08499 5/20 0.53
ACHE P22303 2/20 0.48
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
PPARG P37231 1/20 0.44
PPARD Q03181 1/20 0.44
PPARA Q07869 1/20 0.44
ALDH1A1 P00352 1/20 0.44
CYP2C19 P33261 1/20 0.44
POLB P06746 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1370408 0.87 GAA (0.55) GAATNFPDE4APDE4BPDE4C
SCHEMBL8358428 0.86 GAA (0.50) GAATNFPDE4APDE4BPDE4C
SCHEMBL7363845 0.85 PDE4A (0.61) GAAPDE4APDE4BPDE4CPDE4D
Hydrochloric Acid SCHEMBL11461220 0.85 GAA (0.80) GAATNFPDE4APDE4BPDE4C
SCHEMBL6251186 0.82 TNF (0.55) TNFPDE4APDE4BPDE4CPDE4D
SCHEMBL2987068 0.82 TNF (0.55) TNFPDE4APDE4BPDE4CPDE4D
SCHEMBL5941271 0.82 TNF (0.55) TNFPDE4APDE4BPDE4CPDE4D
Hydrochloric Acid SCHEMBL5743883 0.81 TNF (0.54) TNFPDE4APDE4BPDE4CPDE4D
SCHEMBL8771052 0.80 TNF (0.56) TNFPDE4APDE4BPDE4CPDE4D
SCHEMBL8903093 0.79 GAA (0.46) GAATNFALDH1A1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0584208-A4 1994-03-23 EP disclosed
EP-0584208-A1 PYRROLIDINONES SMITHKLINE BEECHAM CORPORATION (US) 1994-03-02 EP disclosed
WO-1992019594-A1 PYRROLIDINONES SMITHKLINE BEECHAM CORPORATION (US) 1992-11-12 WO disclosed