SCHEMBL7363973

SCHEMBL7363973

O=c1c2cccnc2c(-c2cccc(Br)c2)nn1-c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 3/20 0.50
ALDH1A1 P00352 3/20 0.50
LMNA P02545 2/20 0.50
PDE4A P27815 5/20 0.45
PDE4B Q07343 3/20 0.45
PDE4C Q08493 3/20 0.45
PDE4D Q08499 3/20 0.45
PDE3B Q13370 1/20 0.45
PDE3A Q14432 1/20 0.45
GAA P10253 2/20 0.44
HTT P42858 2/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
CNR1 P21554 1/20 0.43
CNR2 P34972 1/20 0.43
GPR55 Q9Y2T6 1/20 0.43
KDM4E B2RXH2 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7368041 0.91 NPSR1 (0.50) NPSR1ALDH1A1LMNAPDE4APDE4B
SCHEMBL9172942 0.90 NPSR1 (0.45) NPSR1ALDH1A1LMNAPDE4APDE4B
SCHEMBL9168570 0.87 NPSR1 (0.56) NPSR1ALDH1A1LMNAPDE4APDE4B
SCHEMBL7359405 0.86 PDE4A (0.61) NPSR1ALDH1A1LMNAPDE4APDE4B
SCHEMBL7367535 0.83 PDE4A (0.53) NPSR1ALDH1A1LMNAPDE4APDE4B
SCHEMBL9171807 0.83 NPSR1 (0.75) NPSR1ALDH1A1LMNAPDE4APDE4B
SCHEMBL7362724 0.82 PDE4D (0.63) NPSR1ALDH1A1LMNAPDE4APDE4B
SCHEMBL7365641 0.81 PDE4A (0.67) NPSR1ALDH1A1LMNAPDE4APDE4B
SCHEMBL9165717 0.80 NPSR1 (0.61) NPSR1ALDH1A1LMNAPDE4APDE4B
SCHEMBL7363279 0.79 GRM5 (0.48) NPSR1ALDH1A1LMNAPDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0612321-A1 PYRIDO PYRIDAZINONE AND PYRIDAZINTHIONE COMPOUNDS WITH PDE IV INHIBITING ACTIVITY SYNTEX (U.S.A.) INC. (US) 1994-08-31 EP disclosed
WO-1993007146-A1 BENZO AND PYRIDO PYRIDAZINONE AND PYRIDAZINTHIONE COMPOUNDS WITH PDE IV INHIBITING ACTIVITY SYNTEX (U.S.A.) INC. (US) 1993-04-15 WO disclosed